PROGRAM
of the Conference
 
III International Conference on the Chemistry and Biological Activity
of Nitrogen-Containing Heterocycles
June 20–23 2006
(Chernogolovka Research Center, Moscow Region, Russia)
 

 
Monday, June 19, 2006

16:00–21:00 Registration (The Hotel of the Chernogolovka Research Center)

Registration of participants of the conference will be held in the Lobby of the Hotel of the Chernogolovka Research Center.

All participants of the conference should have passports.


Tuesday, June 20, 2006

08:00 Registration (The Foyer of the Conference Hall, the House of Scientists)
 
08:30 Breakfast
 
09:00 Opening Ceremony (The Conference Hall, the House of Scientists)
Opening Keynote Address by Prof. Victor G. Kartsev, Chairman of Organizing committee,
Chairman of "Scientific Partnership" Foundation
 
Greetings by honorary delegates of the conference
 
09:30 Presentation ceremony of the Medal "In memory of Professor A.N. Kost"
and the International ScientificPartnership Foundation's awards

 
Scientific Program


Session I                      Chemistry of synthetic and natural heterocycles


Keynote Lectures

Session Chairpersons: Prof. J. Bergman, Prof. S. Abu-Orabi 

10:30–11:00
 Mąkosza M. (Poland)
Synthesis of indoles via nucleophilic substitution of hydrogen in nitroarenes
11:00–11:40
 Van der Plas H.C. (The Netherlands)
The ring transformation as methodology for the synthesis of azaheterocycles

 
11:40–12:10 Coffee Break (The Lobby of the Conference Hall, the House of Scientists)


Plenary Lectures

Session Chairpersons: Prof. Henk C. van der Plas, Prof. U. Jordis

12:10–12:35
 Bergman J., Stensland B. (Sweden)
Novel syntheses of indoles and related heterocycles
12:35–13:00
 Kartsev V.G. (Russia)
New horizons for use of T-reactions in the synthesis of heterocycles
13:00–13:25
 Preobrazhenskaya M.N. (Russia)
Chemistry and biology of ascorbigen
13:25–13:50
 Vasilevsky S.F., Balova I.A. (Russia)
New one-pot synthesis and heterocyclization of vic-functionalized aryl(hetaryl)alkadiynes-1,3
 

14:00–15:50 Lunch (Restaurant)
 

Session I                      Chemistry of synthetic and natural heterocycles 


Plenary Lectures

Session Chairpersons: Prof. M. Mąkosza, Prof. M. Preobrazhenskaya
 
16:00–16:25
 Fišera L. (Slovak Republic)
Control of regio- and stereoselectivity in nitrone cycloadditions and their utilization in synthesis
16:25–16:50
 Jordis U. (Austria)
How to use software and integrate databases in the daily practice of heterocyclic chemist
16:50–17:15
 Hajós Gy. (Hungary)
Zwitter-ionic heterocycles: A pool of novel polyfused ring systems
17:15–17:40
 Zefirov N.S. (Russia)
Organic chemistry and mathematics: Design and modeling
17:40–18:05
 Dondoni A., Massi A. (Italy)
Multicomponent synthetic approach to reengineered N-heterocycle pharmacophores by glycoside decoration


Oral Presentations

Session Chairpersons: Prof. L. Fišera, Prof. A. Dondoni

18:05–18:25
 Nosova E.V., Lipunova G.N., Laeva A.A., Charushin V.N. (Russia)
Fluorinated 2-substituted [1,3]benzothiazinones: Synthesis and properties
18:25–18:45
 Danagulyan G.G. (Armenia)
Kost–Sagitullin rearrangement with amine exchange and concurrent recyclization of pyrimidinium salts
18:45–19:00
 Aripova S.F., Zhalolov I.Zh., Levkovich M.G., Tashkhodzhaev B.,
Khuzhaev V.U., Mirzaev Yu.R. (Uzbekistan)
New alkaloids from Arundo donax L. for medicinal applications
 
 
14:00–15:50 Poster Session 1 (poster nos. 1–75) (The Lobby of the Assembly Hall,
the Big Reception-Room)
 
Poster nos.
Poster Details

1

 Aboskalova N.I., Smirnova N.N., Skobeleva A.V., Berestovitskaya V.M.
Synthesis of substituted pyrazoles and isoxazoles from gem-acylnitroethenes

2

 Abramov I.G., Voron'ko M.N., Sapegin A.V., Zeifman A.A., Bukhreev P.B., Plakhtinskii V.V.
Phthalonitriles condensed with cycloaliphatic diamines: Synthesis and functionalization

3

 Afon'kin A.A., Kostrikin M.L., Shumeiko A.E., Popov A.F.
6,7-Dimethoxy-1-methyldihydroisoquinoline enamines in reactions of
1,2-cycloaddition

4

 Agedilova Ì.Ò., Turmukhambetov A.Zh., Kazantsev A.V., Adekenov S.M.
Chemical transformations of vasicinone

5

 Akhmedzhanova V.I.
Alkaloids of Haplophyllum perforatum

6

 Akhrem A.A., Baranovskii A.V., Gulyakevich O.V., Mikhal'chuk A.L.
Azangular heterocycles: Structure and molecular dynamics as studied
by high-resolution NMR

7

 Akhrem A.A., Dubovskii V.L., Gulyakevich O.V., Mikhal'chuk A.L., Tikhomirov S.A., Tolstorozhev G.B.
Absorption/emission properties of 3,4-dihydroisoquinolines: Solvation and acid-base interaction with environment

8

 Akhrem A.A., Govorova A.A., Gulyakevich O.V., Lyakhov A.S.,
Mikhal'chuk A.L., Skornyakov I.V., Tolstorozhev G.B.
Intermolecular interactions of immuno-active azasteroids by IR spectroscopy and XRD

9

 Akhrem A.A., Gulyakevich O.V., Govorova A.A., Kurman P.V.,
Lyakhov A.S., Mikhal'chuk A.L.
3-Acetyl-4-methylpyrido[2,1-a]isoquinoline-2-ones.
[2+4]-Cyclocondensation of 3,4-dihydroisoquinolines with triacetylmethane

10

 Akopyan Sh.F.
Pyrimidine derivatives in synthesis of condensed triazolo-, tetrazolo-, and imidazolopyrimidines

11

 Aksenov A.V., Trifonov V.V., Goncharov V.I.
2,3'-Biquinoline derivatives by Vilsmeier reaction

12

 Amiranashvili L.Sh., Merlani M.I.
17-Aza-16,17a-D-homoandrost-2-ene from tigogenine

13

 Andreev G.N., Shults E.E., Tolstikov G.A.
Synthesis of 5,5-cyclofused barbituric acids

14

 Andriyankova L.V., Mal'kina A.G., Nikitina L.P., Trofimov B.A.
Functionalized polyconjugated 1,4-dihydropyridines from pyridine and phenylcyanoacetylene

15

 Angenot L., Akhmedzhanova V.I., Akhmedkhodzhaeva Kh.S.,
Nazrullaev S.S.
Biological activity of alkaloids from plants of the Haplophyllum genus

16

 Anisimova N.A., Ladygin V.V., Berestovitskaya V.M.
Synthesis of functionalized carbazoles

17

 Anisimova V.A., Tolpygin I.E., Askalepova O.I.
Interaction of 2,9-disubstituted imidazo[1,2-a]benzimidazoles
with tetracyanoethylene

18

 Anisimova V.A., Tolpygin I.E., Askalepova O.I.
Synthesis of 2,3-dihydroimidazo- and 2,3,4,10-tetrahydropyrimido-
[1,2-a]benzimidazolyl-N-acetic acids and their derivatives

19

 Arsen'eva M.Yu., Arsen'ev V.G., Minkin V.I.
New derivatives of furo[3',4':3,4]cyclohepta[d]imidazoles

20

 Babakova M.N., Vlaskina N.M., Suzdalev K.F., Mezheritskii V.V.,
Kartsev V.G.
Ò-Reactions in synthesis of condensed a-carbolines

21

 Bakbardina O.V., Pukhnyarskaya I.Yu., Fazylov S.D., Gazaliev A.M.
Potassium b-aminoethylxanthogenates from alkaloids

22

 Bakbardina O.V., Rakhimzhanova N.Zh., Gazaliev A.M., Fazylov S.D.
New carbamoyloxamidinesfrom anabasine and cytosine

23

 Bakharev V.V., Gidaspov A.A.
Alkylation of 5-trinitromethyltetrazolo[1,5-a]-1,3,5-triazine salts

24

 Bannikova Yu.N., Khalturina V.V., Sedegova E.A., Maslivets À.N.
Heterocyclization of 2,3-dihydro-2,3-pyrrolediones under the action
of binucleophiles

25

 Bauman V.T., Shults E.E., Tolstikov G.A.
Synthesis of C(1)-substituted pyrrolidinothebaines

26

 Begunov R.S., Ryzvanovich G.A., Nozdracheva O.I.
Condensed pyridines containing a central nitrogen atom

27

 Belov E.Yu., Tomachinskii S.N., Dybenko A.G.
Amino-acid modification of spinaceamine

28

 Belyuga A.G., Balya A.G., Brovarets V.S.
Recyclization of 4-acylamino-5-aryl-2-phenacylthio-1,3-oxazoles upon heating in polyphosphorous acid

29

 Biitseva À.V., Gordienko Î.V., Kornilov Ì.Yu., Sukach V.À., Vovk Ì.V.
Regioselective cyclocondensation of 1-arylimino-1Í-isoindole-3-amines with a-chlorobenzyl isocyanates

30

 Bilokin' M.D., Pivovarenko O.V., Yushchenko D.A., Duportail G., Mely Y., Pivovarenko V.G.
New derivatives of 3-hydroxyquinolone: Dyes displaying two-band fluorescence

31

 Boldashevskii A.V., Ibraev M.K., Fazylov S.D., Gazaliev A.M., Nukhuly A.
bis-Thioethers from alkaloids and their analogs

32

 Bondarenko S.P., Frasinyuk M.S., Khilya V.P.
Heteroanalogs of isoflavone in reaction with hydroxylamine

33

 Borisova Yu.Yu., Mironov V.F., Burnaeva L.A., Amerkhanova N.K., Konovalova I.V.
Nitrogen-containing heterocycles from phosphorylated derivatives of hydroxynicotinic acid

34

 Borisova Yu.Yu., Mironov V.F., Burnaeva L.A., Amerkhanova N.K., Konovalova I.V.
Reactions of 2-R-benzo[d]-1,3,2-oxazaphosphorin-6-ones with compounds containing activated multiple bonds

35

 Borovik V.P., Shkurko O.P.
2-Thio derivatives of 4-phenyl-9H-pyrimido[4,5-b]indole

36

 Bulychev Yu.N., Bakharev V.V., Gidaspov A.A.
Cytotoxic activity of 2-R1-4-R2-6-trinitromethyl-1,3,5-triazines

37

 Bulychev Yu.N., Bakharev V.V., Gidaspov A.A.
Cytotoxic activity of 3,4-di(2'-R1-4'-R2-1,3,5-triazin-6'-yl)-1,2,5-oxadiazole-N-oxides

38

 Butov G.M., Parshin G.U., Panyushkina O.A., Mokhov V.M.
New methods for synthesis of (1-adamantyl)azoles

39

 Buzykin B.I., Kovalenko V.I., Ginzburg B.M., Nurgatin V.V.
1,4,5,8,9,10-Hexaazaperhydrodiethano[4,9][8,10]anthracene

40

 Bykov E.E., Lakatosh S.A., Preobrazhenskaya M.N.
Reaction of bisindolylmaleimides with protic acids: Quantum-chemical study

41

 Bykova V.V., Usol'tseva N.V., Anan'eva G.A., Znoiko S.A., Maizlish V.E., Shaposhnikov G.P.
Copper phthalocyanines containing benzotriazole fragments: Synthesis and mesomorphism

42

 Chesnyuk A.A., Mikhailichenko S.N., Zaplishnyi V.N., Neshchadim N.N., Konyushkin L.D.
A new conjugated heterocyclic system, 2-(1-pyrrolyl)-4,6-disubstituted 1,3,5-triazine

43

 Chikvaidze I.Sh., Samsoniya Sh.A., Targamadze N.L., Samsonia N.Sh., Kalatozishvili A.Z., Narimanidze N.O., Barbakadze N.N.
New polycyclic heterocycles containing indole and pyridazine moieties

44

 Chukhajian E.O., Nalbandyan M.K., Gevorkyan H.R., Khachatryan À.À.
Intramolecular recyclization of isoindolinium salts and their condensed analogs

45

 Churikov D.G., Kulinkovich O.G.
Transformation of carboxylic esters into 5-substituted isoxazoles

46

 Dabaeva W.W., Bagdasaryan M.P., Noravyan A.S.
1-Amino-3H-6,6,7-trimethylpyrazolo[3,4-b]-
5,6,7,8-tetrahydro[1,6]naphthyridine dihydrochloride: Synthesis and
anti-monoaminooxydase effect

47

 Danagulyan G.G., Boyakhchyan A.P., Sahakyan L.G., Danagulyan A.G.
Synthesis and recyclization of some azolo[1,5-a]pyrimidines

48

 Danagulyan G.G., Tadevosyan D.A., Hakobyan V.P., Balasanyan M.G., Ashrafyan K.B.
Synthesis and cerebrovascular activity of some pyrazolo[1,5-a]pyrimidines

49

 Deev S.L., Rusinov V.L., Ulomskii E.N., Shestakova T.S., Chupakhin O.N., Kukhanova M.K., Khandazhinskaya A.L., Shirokova E.A.
Abnormal nucleosides from 1,2,4-triazolo[5,1-c][1,2,4]triazin-7-ones

50

 Demidchuk B.A., Brovarets V.S., Chernega A.N.
Cyclocondensation of 1-aryl-1,3,4,4-tetrachloro-2-aza-1,3-butadienes with
2-aminobenzimidazole and its homologs

51

 Detistov A.S., Zaremba O.V., Kovalenko S.N.
Combinatorial library of 5-(5-methyl-1H-1,2,3-triazol-4-yl)-
1,2,4-oxadiazoles

52

 Dimukhametov M.N., Abdrakhmanova L.M., Mironov V.F., Ivkova G.A., Zagidullina E.R., Musin R.Z.
5,7-Dioxa-1-aza-6-phospha-benzo[3,4]bicyclo[4,3,1]decane-2,6-diones through intramolecular cycle expansion in
2-benzylideneàminoethyl(phenyl) salicyl phosphites

53

 Dimukhametov M.N., Mironov V.F., Abdrakhmanova L.Ì., Musin R.Z.
Reaction of iminophenols with chlorophosphites as a new route to
N,P-containing màcroheterocycles

54

 Dmitriev A.S., Abaev V.T., Pilipenko A.S., Podelyakin S.A., Gavrilov À.À., Butin À.V.
Amides of o-carboxybenzylfuran in synthesis of isoquinolone derivatives

55

 Dmitrieva I.G., Dyadyuchenko L.V., Kaigorodova E.A.
4,6-Dimethyl-5-R-3-cyanopyridyl-2-sulfonyl chlorides

56

 Dotsenko V.V., Krivokolysko S.G., Litvinov V.P.
New derivatives of pyridin-4(1H)-one from diketene and cyanothioacetamide

57

 Dubovik I.P., Garazd Ì.Ì., Vinogradova V.I., Khilya V.P.
Modification of cytisine with coumarinyloxyacetic acids

58

 Dyachenko V.D.
cross-Recyclizationof4-alkyl(aryl, heteryl)-2,6-diamino-3,5-dicyano-
4H-thio(seleno)pyrans

59

 Dybenko A.G., Yazlovitskii A.V., Patrikei S.Yu.
New peptoids bearing a heterocyclic fragment

60

 Dzhavakhishvili S.G., Gorobets N.Yu., Paponov B.V., Desenko S.M.
Transformations of Gewald amides in their reactions with aldehydes

61

 Egamov D.I., Yakubov U.M., Shakhidoyatov Kh.M.
Reaction of quinazolone thioimidium salts with aromatic amines

62

 Elmuradov B.Zh., Shakhidoyatov Kh.M.
O-Alkyl derivatives of quinazoline alkaloids

63

 Elmuradov B.Zh., Shakhidoyatov Kh.M.
Reaction of α-oxymethylidene-2,3,4,10-tetrahydro-1H-pyrido-
[2,1-b]-quinazolin-10-one with anabasine and cytisine

64

 Elmuradov B.Zh., Turdibaev Zh.E., Shakhidoyatov Kh.M.
a-Piperazinylmethylidene derivatives of quinazoline alkaloids

65

 Eshmatov A.K., Topchieva T.S., Andreev S.A., Tashmukhamedova À.K.
Phenazine derivatives from dibenzo-18-crown-6

66

 Fedorova O.V., Zhidovinova M.S., Ovchinnikova I.G, Valova M.S.,
Kharchuk V.G, Rusinov G.L.
New approaches to multicomponent synthesis of azaheterocycles and heterocycle-containing podands

67

 Frasinyuk M.S., Khilya V.P.
Aminomethylation of 2-amino-3-(2-benzothiazolyl)chromones

68

 Frolov K.À., Dotsenko V.V., Krivokolysko S.G., Litvinov V.P.
New tetrahydronicotineamide derivatives

69

 Frolov K.À., Dotsenko V.V., Krivokolysko S.G., Litvinov V.P.
Reduction of (Å)-3-aryl-2-(thiazole-2-yl)acrylonitriles with LiAlH4

70

 Gabrielyan S.H., Markosyan A.I.
Some transformations of 3-furfuryl-4-oxo-2-thioxo-
1,2,3,4,5,6-hexahydrospiro(benzo[h]quinazoline-5,1'-cyclohexane)

71

 Gazaliev A.M., Nurkenov O.A., Adambekova K.A.
Synthesis of 2-(N-diethylthiocarbamoylthio)-3,4-dimethyl-5-phenyl-
1,3,2-oxazîphospholanes

72

 Gazaliev A.M., Nurkenov O.A., Aynabaev A.A., Bessonov D.V., Ermukhanbetova R.A.
Chemical modification of some N-xylosyl- and N-glycosylamines

73

 Gazaliev A.M., Nurkenov O.A., Sultanov A.S., Ibysheva Sh.T.
New oxazolidines from ephedrine alkaloids

74

 Gazieva G.A., Lozhkin P.V., Kravchenko A.N.
Reaction of 4,5-dihydroxyimidazolidin-2-ones with sulfamides

75

 Gidaspov A.A.
Trinitromethylation of 2,4,6-trichloro-1,3,5-triazine in the presence of water, alcohols, and phenols
 
 
19:20–20:30 Welcome Cocktail Party (The Lobby of the Conference Hall, the House of Scientists)
 

Wednesday, June 21, 2006
 
8:30 Breakfast


Session I                      Chemistry of synthetic and natural heterocycles 

Keynote and Plenary Lectures (The Assembly Hall, the Big Reception-Room)

Session Chairpersons: Prof. H.-J. Knölker, Prof. S. Vasilevsky 

9:00–9:30
 Atta-ur-Rahman, Choudhary M.I. (Pakistan)
Nitrogen-containing heterocycles from natural sources: Isolation, biological studies, and synthesis
9:30–9:55
 Florio S. (Italy)
o-Lithiation: a useful strategy towards heterocycles
9:55–10:20
 Chupakhin O.N., Rusinov V.L., Charushin V.N. (Russia)
Abnormal nucleosides from isosteres of purine

Oral Presentation
 
10:20–10:35
 Van der Eycken E. (Belgium)
Microwave irradiation: A 'green tool' in 2(1H)-pyrazinone chemistry

Plenary Lecture 

10:35–11:05
 will be announced later
 
11:10–11:30 CoffeeBreak (The Banquet Hall, the Big Reception-Room)
 
Oral Presentations

Session Chairpersons: Prof. O. Chupakhin, Prof. S. Florio

11:30–12:00
 Agarwal S., Filali S., Fröhner W., Knöll J., Krahl M.P., Reddy K.R.,
Knölker H.-J. (Germany)
Application of oxidative cyclizations to the synthesis of bioactive
nitrogen-containing heterocycles
12:00–12:15
 Abu-Orabi S.T. (Jordan)
Utilization of 1,2,3-dipolar cycloaddition reactions of azides toward
the synthesis of 5-membered rings heterocyclic compounds
12:15–12:30
 Nemes A. (Hungary)
Synthetic studies related to cis- and trans-apovincamine derivatives and metabolites
12:30–13:00
 Rádl S., Klecán O. (Czech Republic)
New approaches to the synthesis of triptans
13:00–13:15
 Bölcskei H., Gács-Baitz E., Szántay Cs. Jr., Kalaus Gy.,
Szántay Cs. (Hungary)
Synthesis of indoloazepines and indoloazocines
13:15–13:30
 Geronikaki A., Incerti M., Zani F., Vicini P. (Greece)
2-Benzo[d]isothiazolylimino-5-arylidene-4-thiazolidinones: Synthesis and antimicrobial activity
13:30–13:45
 Shklyaev Yu.V., Glushkov V.A., Stryapunina O.G., Rozhkova Yu.S.,
El'tsov M.A. (Russia)
The synthesis of partially hydrohenization azine and azole: Dihydroisoquinolines, spiropyrrolines, polyhydroindolines

13:45–15:15 Lunch (Restaurant)
 

Session I                      Chemistry of synthetic and natural heterocycles

Oral Presentations
 
Session Chairpersons: Prof. S. Rádl, Prof. A. Geronikaki

15:15–15:30
 Bazureau J.P., Legeay J.C., Fraga-Dubreuil J., Hakkou H. (France)
Ionic liquid-phase technology: A new tool for combinatorial chemistry. Applications in heterocyclic chemistry mediated by microwave
dielectric heating
15:30–15:45
 Voskressensky L.G., Vorob'ev I.V., Varlamov A.V. (Russia)
Unusual reactions of tetrahydrobenzo[b][1,6]naphthyridines with activated alkynes
15:45–16:00
 Korotkikh N.I., Raenko G.F., Kiselev À.V., Knishevitsky À.V., Shvaika Î.P., Glinyanaya N.V., Panov I.S., Cowley À.H., Jones J.N., Moore J.A. (Ukraine)
Stable carbenes. Insertion into Ñ–Í bonds and reaction with ester function. New cleavage and thermal transformation of 1,2,4-triazol-5-ylidenes
16:00–16:15
 Stroganova T.A., Vasilin V.K., Krapivin G.D. (Russia)
Amino acids of the thieno[2,3-b]pyridine series in reactions of intramolecular cyclization
16:15–16:30
 Gorobets N.Yu., Ermolaev C.A., Dzhavakhishvili S.G., Sirko S.N., Chernenko V.N., Desenko S.M. (Ukraine)
2-Dimethylaminomethylene-1,3-cyclohexanedione derivatives in reaction with methylene-active nitriles
16:30–16:45
 Makhova N.N., Shevtsov A.V., Petukhova V.Yu., Kuznetsov V.V.,
Kislukhin A.A. (Russia)
Transformation of diaziridine ring under the action of ketenes as a new synthetic approach to nitrogen-containing heterocyclic systems
16:45–17:00
 Polygalova N.N., Mikhailovskii A.G., Vakhrin M.I. (Russia)
Carbonyl derivatives of condensed isoquinolines: Synthesis and reactivity
 
17:00–17:20 Coffee Break
 

Oral Presentations

Session Chairpersons:Prof. J.P. Bazureau, Prof. H. Bölcskei, Prof. L. Voskressensky

17:20–17:35
 Suzdalev K.F., Babakova M.N., Den'kina S.V, Kartsev V.G. (Russia)
Indoles bearing reactive groups for synthesis of combinatorial libraries
17:35–17:50
 Vizer S.A., Dedeshko E.H., Erzhanov K.B., Dembitskii V.M. (Kazakhstan)
Synthesis of N-containing heterocycles from a-propargyl-b-dicarbonyls and their O-phosphoryl derivatives
17:50–18:05
 Lesyk R.B., Zimenkovsky B.S., Atamanyuk D.V. (Ukraine)
Thiopyrano[2,3-d]thiazoles and their derivatives: Synthesis and biological activity
18:05–18:20
 Kozminykh V.O., Goncharov V.I., Kozminykh E.N., Fiergang S.I. (Russia)
Synthesis of oxoalkylidene(oxocycloalkyl)quinoxalinones


Session II   Biological activity of nitrogen-containing heterocycles
(Lecture-Room 2, The Big Reception-Room)

Plenary Lectures
  
Session Chairpersons: Prof. N. Zefirov, Prof. À. Saxena, Prof. V. Poroikov

15:00–15:25
 Zefirov N. (Russia)
The use of QSAR in the search of biologically active compounds
15:25–15:50
 Poroikov V.V., Filimonov D.A., Gloriozova T.A., Lagunin A.A. (Russia)
Computer-aided prediction of biological activity for nitrogen-containing organic compounds
15:50–16:15
 Saxena À. (India)
Substituted arylpiperazines in rational drug design

Oral Presentations
 
16:15–16:30
 Mali A., Shelar M., Shelar A. (India)
Antibiotic resistance: A search for new b-lactam antibiotics
16:30–16:45
 Chung M.C. (Brazil)
Prodrug design: Improving drug activity
16:45–17:00
 Belous A.R. (USA)
Endogenous indole compounds: biological significance of
5-hydroxytriptamine and its metabolites
 
17:00–17:20 Coffee Break

 
Oral Presentations
 
17:20–17:35
 Granzhan A., Ihmels H., Viola G. (Germany)
Rearrangements in diazoniapentaphenes and DNA-binding properties
of diazoniapolycycles
17:35–17:50
 Duburs G., Bisenieks E., Krauze A., Plotniece A., Sobolevs A., Tirzitis G., Vigante B. (Latvia)
Dihydropyridine derivatives as biomimetics and bioprotectors
17:50–18:05
 Veinberg G., Vorona M., Shestakova I., Kanepe I., Lukevics E. (Latvia)
Antitumor 3a-chloro- and 3-alkylideneazetidinone-2 derivatives

 
9:00–19:00  Poster Session 2 (poster nos. 76–150) (The Lobby of the Assembly Hall,
the Big Reception-Room)
 
Poster nos.
Poster Details

76

 Gladkov E.S., Desenko S.M., Sirko S.N.
Three-component cyclocondensation of aminoazoles with cyclic ketosulfones and aldehydes

77

 Gorbulenko N.V., Kurdyukova I.V., Turov À.V., Khilya V.P.
2-Aminoimidazo[1,5-a]pyrimido[5,4-c]quinolin-10-ol as a new condensed heterocyclic system

78

 Gorbulenko N.V., Tkachuk Ò.M., Shokol Ò.V., Semenyuchenko V.V.,
Khilya V.P.
Annelation of oxazine cycle to 3-hetarylchromones through Mannich's reaction

79

 Gorichko M.V., Komarov I.V., Patrikei S.Yu.
Conformationally rigid analogs of cyclic a-amino acids

80

 Gulyakevich O.V., Mikhal'chuk A.L., Akhrem A.A.
[2+4]-Cyclocondensation of cyclic Schiff bases with b-di-, b,b'-tricarbonyl compounds: Perycyclic heterocyclization of iminium cations with enol anions of b-di-, b,b'-tricarbonyl compounds

81

 Gusakova N.V., Shikhaliev Kh.S., Shestakov A.S.
Regioisomeric pyrazoles from 4,6-dimethylpyrimidinyl-2-hydrazine and esters of 3-oxoacids

82

 Ibraev Ì.K., Kîzhinà Zh.Ì., Gàzàliev À.M., Fazylov S.D., Takibaeva A.T.
N-[(5-thioxo-4,5-dihydro-1,3,4-oxa-diazol-2-yl)methyl]benzamides

83

 Ibragimov Ò.F., Saprykina V.A., Shakhidoyatov Kh.M.
Condensation of heterocyclic amines with N-methylol lactams

84

 Isaikina O.G., Kalinin A.A., Mamedov V.A.
Tiazolo[3,4-a]quinoxaline monopodands from
bis-3-(a-bromoethyl)quinoxalin-2-ones and thiourea

85

 Ishchenko V.V., Shablykina O.V., Shablykin O.V., Khilya V.P.
3-Hetarylisocoumarins: Synthesis and transformation into
3-hetarylisoquinolones

86

 Ivanov S.P., Nugumanov T.R., Spirikhin L.V., Murinov Yu.I.
4-Methyl-5-hydroxyuric acid from 5-hydroxy-6-methyluracil
in aqueous solution

87

 Ivkova G.A., Mironov V.F., Burnaeva L.M., Konovalova I.V.,
Shemetova A.S., Ogurtsova E.V.
2,5-Dioxobenzo[f]-1,4,2-oxazaphosphepines by reaction of 3-alkyliminopyridines with salicylphosphites

88

 Kagarlitskii A.D., Balpanov D.S., Krichevskii L.A., Postnikov L.S.
Oxidative ammonolysis of 2-methyl-3-hydroxyquinoxaline

89

 Kalinichenko Å.N., Zhernosek Å.V., Litvinko N.Ì., Kuchuro S.V.,
Rakhuba G.N.
2',3'-Dideoxycytidine-5'-monophosphate-phosphatidylethanolamine-phosphoramidate: Synthesis and interaction with phospholipase À2

90

 Kartsev V.G., Serov A.B., Sukhotin A.V.
New derivatives of couroupitine A (tryptanthrine): Synthesis and transformations

91

 Kas'yan L.I., Karpenko D.V., Kas'yan A.O.
Reaction of norbornene sulfonamides with organic peracids

92

 Katorov D.V., Illarionova T.A., Rudakov G.F., Zhilin V.F.
Synthesis of heterocyclic geminal nitroazides

93

 Khilya O.V., Vintonyak V.V., Volovenko Yu.M.
Reaction of hetarylacetonitriles with heterocyclic 1,3-bielectrophilic halocarbonyls

94

 Khudina O.G., Shchegol'kov E.V., Burgart Y.V., Saloutin V.I.
Ring–chain transformations of 7-fluoroalkyl-4,7-dihydroazolo[5,1-c]triazines in reaction with hydrazides and thiosemicarbazide

95

 Kislukhin À.À, Shevtsov À.V., Kuznetsov V.V., Makhova N.N.
N-acyl- and N,N-bisacylpyrazolidines from 1,5-diazabicyclo[3,1,0]hexanes and acyl chlorides

96

 Kolobov A.V., Panfilov S.T., Borisov P.V., Kofanov E.R.
Arylpyridazines: Synthesis, structure, chemical behavior

97

 Kol'tsov N.Yu.
Reduction of heterocyclic a-aminonitriles with lithium aluminum hydride

98

 Komykhov S.A., Petrova M.G., Borovskoi V.A., Musatov V.I.,
Desenko S.M.
New dihydropyrazolo[1,5‑a]pyrimidine derivatives  by three-component condensation of 3-aminopyrazole-4‑arylcarboxamides with carbonyls

99

 Kopteva N.I., Stepanova T.V.
Heterocyclization of coumarin-3-carboxylic acid hydrazide

100

 Korotkikh N.I., Kiselev À.V., Kovalenko A.N., Shvaika O.P., Cowley À.H., Jones J.N., Moore J.A.
New routes to synthesis of carbene complexes with alkali and transition metals from heteroaromatic carbenes and their precursors

101

 Koshchienko Yu.V.
Synthesis of dihetarylphenylcarbinols involving organometallic compounds

102

 Kostenev I.S., Ovcharov M.V., Voskressensky L.G., Varlamov A.V.
Heteroannelated pyridopyrimidines: Synthesis and transformations

103

 Kostenko E.S., Kaigorodova E.A., Krapivin G.D.
4-(3-Pyridyl)-1,6-dihydro-6-pyrimidinones

104

 Kostrub V.V., Shevchenko M.A., Tsupak E.B.
Pyrimido[d]pyriliuim salts in synthesis of new fused nitrogen-containing heterocycles

105

 Kovalenko S.N., Vlasov S.V., Silin A.V., Chernykh V.P.
Reaction of 2-iminocoumarin-3-carboxamides with 2-aminothiobenzamide

106

 Krasnov V.P., Levit G.L., Zhdanova E.A., Solieva N.Z., Sadretdinova L.Sh., Chupakhin O.N.
Kinetic resolution of racemic piperidine derivatives

107

 Kryl'skii D.V., Shikhaliev Kh.S., Didenko V.V.
Heterocyclic systems from aminopyrazoles and diketones

108

 Kryl'skii D.V., Shikhaliev Kh.S., Didenko V.V.
Pyrazolotriazines from aminopyrazoles and ÑÍ-active compounds

109

 Krysin M.Yu., Petrov V.V., Muratov D.N.
Indeno[1,2-d]pyrimidines from 2-arylidene-1,3-indandiones and guanidines

110

 Kurbatov E.S., Krasnikov V.V., Pavlenko D.A., Mezheritskii V.V.
Rearrangement of pyrano[2,3-d]pyrimidines

111

 Kurbatov S.V., Goumont R., Tatarov A.V., Terrier F.
Functionalization of nitrobenzodifuroxan with dienes generated in situ

112

 Kutrov G.P., Kovalenko N.V., Cherepakha A.Yu.
Reaction of heterocyclic imidazo bromides with oxidizers

113

 Kuznetsov A.Yu., Kholopov U.A., Chapyshev S.V., Nam N.L.
2-Piperidine-substituted 4-aminopyrimidines by reduction of
4-amino-2-pyridylpyrimidines

114

 Kuznetsov A.Yu., Kholopov U.A., Chapyshev S.V., Nam N.L.
New 5,6,7,8-tetrahydropyrido[d]pyrimidines

115

 Kuznetsov D.V., Neskubo A.A., Andreev S.A., Tashmukhamedova A.K.
2-Amino-5-(-dibenzo-18-crown-6-yl)-thiadiazole

116

 Kuznetsov V.V., Makhova N.N.
New stable heterocyclic a-hydroxy-N-chloroalkylamines

117

 Kuznetsov V.V., Makhova N.N., Terpigorev A.N.
New method for synthesis of alkyl-substituted diaziridines

118

 Kîtovskaya S.K., Tzoi Å., Charushin V.N.
Fluorinated 3,8-dihydroxyquinolines, analogs of natural antitumor
drug Jeneol

119

 Kîtovskaya S.K., Zhumabaeva G.À., Perova N.Ì., Chupakhin O.N., Charushin V.N.
Tandem SNH(AO) and SNipso(AE) reactions in synthesis of fluorinated 3-amino-1,2,4-benzotriazines

120

 Lapteva E.S., Kayukova O.V., Kayukov Ya.S., Ershov O.V.
Substituted 6,6-(2-oxoindol-3,3-ylidene)-3-azabicyclo[3,1,0]hexane-
1,5-dicarbonitriles

121

 Levinson F.S., Akimova S.A., Khasanov R.Kh., Sharnin G.P., Efimov S.I., Falyakhov I.F., Ermolaeva E.A., Varganov R.V., Vasyutina E.A.,
Shakirova I.M.
Nitroso- and nitrosonitrohalonitriles in synthesis of 4,6-dichloro- and
4-methoxy-6-chloro-5,7-dinitrofurazan

122

 Levinson F.S., Ermolaeva E.A., Kalimullina N.I., Vasyutina E.A.,
Varganov R.V.
4-Aminobenzofurazans containing residua of secondary amines

123

 Levinson F.S., Khasanov R.Kh., Sharnin G.P., Gafarov A.N.
Bromonitrobenzofurazans in the Ullmann reaction

124

 Levkovich M.G., Proskurina U.G.
Effect of solvent on chemical shifts in 1H NMR spectra of alkaloids

125

 Levov N.N., Le Tuan Anh, Komarova A.I., Gimranova G.S., Soldatova S.A., Soldatenkov A.T.
Diarenopiperidinomonoaza-14-crowno-4-phanes: Synthesis and reactions

126

 Mamedov V.A., Khafizova E.A., Beschastnova T.N., Rizvanov I.Kh., Berdnikov E.A.
Three-component condensation of pyrid-2-one with bis-(2-chloroethyl)amine hydrochloride as a new method for oxazolidinoethylation

127

 Mamedov V.A., Khafizova E.A.
Chelate azolo[a]annelated qunoxalines from phenylhalopyruvates and their structural analogs

128

 Marakhovskaya T.G., Shchurova N.A., Tyrkov A.G.
New functionally modified 1,2,3-triazoles based on 5-nitromethyl-
1,2,4-oxadiazoles

129

 Markosyan A.I., Dilanyan S.V., Arsenyan F.H., Sukasyan R.S., Garibdzhanyan B.T.
Benzo[h]quinazolines from 1-amino-3-ethyl-3-methyl-2-cyano-
3,4-dihydronaphthalene

130

 Maslivets À.N., Racheva N.L., Shklyaev Yu.V.
Functionalized spiro-bis-heterocyclic systems

131

 Matiichuk V.S., Gorak Yu.I., Lytvyn R.Z., Obushak M.D.
Cyclization of 2-àcyl-5-arylfurans

132

 Medvedeva S.M., Shikhaliev Kh.S., Solov'ev A.S.
New derivatives of spiro-b-carbolines

133

 Mel'chin V.V., Butin A.V.
2-Arylfurans in synthesis of indole derivatives

134

 Melekhin E.A., Bardasov I.N., Ershov O.V., Kayukov Ya.S.
2,4-Diamino-7-hydroxy-10-aryl-10Í-9-oxa-1-azaanthracene-3-carbonitrile

135

 Melekhin E.A., Bardasov I.N., Ershov O.V., Kayukov Ya.S.
10-R-5-Aryl-2,4-diamino-8,8-dimethyl-6-oxo-
5,6,7,8,9,10-hexahydrobenzo[b]-1,8-naphthyridine-3-carbonitriles

136

 Mel'nikov V.V., Il'ina I.G., Ivanov A.A., Tarasevich B.N.
Autocomplexes of the nitroquinoline series: Synthesis and
spectral investigation

137

 Merlani M.I., Amiranashvili L.Sh., Davitishvili M.G.
Ketosteroid hydrazones: Synthesis and bioactivity

138

 Mishchenko D.V., Frog E.S., Finegold I.I., Kotel'nikova R.A.,
Bogdanov G.N.
2,4,6-Trimethyl-3-oxypyridine nitrosuccinate as a membranoprotector
at oxidative stress

139

 Moiseev S.V., Cherstkov V.F., Vasil'ev N.V.
Synthesis and cycloaddition reactions of polyfluorinated imines and ketones

140

 Mol'kov S.N., Eremkin A.V., Ershov O.V.
2-(3-Amino-8-R-1,4-diazaspiro[4,5]dec-3-en-2-ylidene) malonodinitriles

141

 Mol'kov S.N., Eremkin A.V., Ershov O.V., Kayukov Yu.S.
5,5,6-Trialkyl-2-halo-6-hydroxy-5,6-dihydro-3,4,4(1í)-pyridinetricarbo­nitriles 5,6-Dialkyl-2-halo-3,4-pyridinedicarbonitriles

142

 Mostovaya O.A., Shakirova E.R., Khusainova N.G., Cherkasov R.A.
Reaction of 2H-1,2,3-diazaphosphole with pyrocatechol

143

 Mukusheva G.K., Turmukhambetov A.Zh., Kazantsev A.V., Adekenov S.M.
Aminomethylation of glaucine

144

 Murav'eva E.A., Chebanov V.A., Musatov V.I., Desenko S.M.
Ultrasound-activated synthesis of 2,4,6-tri- and 2,2,4,6-tetra-substituted 1,2,5,6-tetrahydropyrimidines

145

 Musina L.A., Shults E.E., Tolstikov G.A., Adekenov S.M.
Synthesis of substituted indolizines

146

 Nagorichna I.V., Garazd Ì.Ì., Garazd Ya.L., Khilya V.P.,
Ogorodniichuk A.S.
Synthesis of linear and angular pyranodihydrobenzoxazines

147

 Nekrasov D.D., Obukhova A.S., Kharitonova A.V., Khlåbnikova Ò.B.
Stereoisomeric 6-aryl-2-(2-thienyl)-3-(abieta-8,11,13-trien-18-yl)-
1,3-îxazin-4-înes

148

 Nevolina T.A., Shevlyakov M.V., Stroganova T.A.
Amines of the furan series in synthesis of nitrogen-containing heterocycles

149

 Nurmagambetov Zh.S., Turmukhambetov A.Zh., Serperov K.S.,
Kazantsev A.V., Adekenov S.M.
Halogenation of stachydrine

150

 Oganisyan Art.Sh., Oganisyan A.Sh., Noravyan A.S.
4,7,7-Substituted pyrano[4',3':4,5]thienoimidazo[1,2-a]pyrimidine-5-diones
 
20:00  Banquet
 
 
Thursday, June 22, 2006
(For Foreign Delegates)

08:00–09:00 Breakfast
9:00–14:00 Social events for foreign guests (sightseeing tour of Moscow, the Kremlin, a visit to the Cathedral of Christ-the-Savior, entertainment program)
14:00–15:00 Lunch
15:00–20:00  Cultural program continued
 
21:00   Snacks & wine party
 
 
Thursday, June 22, 2006
(Session For Russian and CIS Delegates. Working language is Russian)
(The Assembly Hall, the Big Reception-Room)
 
08:00–09:00 Breakfast
 

Session I                      Chemistry of synthetic and natural heterocycles
 
Plenary Lectures 

Session Chairpersons: Prof. Yu. Shklyaev, Prof. L. Gornostaev

9:00–9:25
 Tolstikov G.A. (Russia)
Synthetic transformation of morphinane and diterpene alkaloids
9:25–9:50
 Granik V.G. (Russia)
Biotransformations of heterocyclic nitrogen-containing drugs
9:50–10:15
 Sagitullina G.P., Sagitullin R.S. (Russia)
Recyclization of pyridinium salts: New horizons
10:15–10:40
 Akhrem A.A., Gulyakevich O.V., Mikhal'chuk A.L. (Belarus)
[2+4]-Cyclocondensation of monocyclic azomethines with b-di- and
b,b'-tricarbonyl compounds in synthesis of azangular heterocycles
10:40–11:05
 Kostyanovsky R.G. (Russia)
Nitrogen chirality in heterocyclic chemistry
11:05–11:30
 Shestopalov A.M., Rodinovskaya L.A., Shestopalov A.A. (Russia)
Recyclization reactions of degenerate carbo- and heterocycles: Practical retrosynthetic approach to new multicomponent methods for synthesis
of N-containing five- and six-membered heterocycles
11:30–11:55
 Saloutin V.I., Burgart Ya.V., Chupakhin O.N. (Russia)
Design of azaheterocycles based on fluorine-containing 2,4-dioxobutanoates and their derivatives
 
12:00–12:20 CoffeeBreak (The Banquet Hall, the Big Reception-Room)
 

Oral Presentations

Session Chairpersons: Prof. G. Tolstikov, Prof. V. Granik

12:20–12:35
 Drach B.S., Sviripa V.N., Pil'o S.G., Popil'nichenko S.V., Golovchenko A.V., Brovarets V.S. (Ukraine)
Synthesis of functionalized condensed heterocycles from 2-acylamino-
3,3-dichloroacrylonitriles
12:35–12:50
 Velikorodov À.V. (Russia)
Quinones and quinoids in synthesis and modification of indoles
12:50–13:05
 Adekenov S.Ì. (Kazakhstan)
Nitrogen-containing derivatives of natural sesquiterpene lactones
13:05–13:20
 Berestovitskaya V.M., Anisimova N.A., Makarova N.G. (Russia)
Synthesis of nitrogen-containing heterocycles from
b-nitroethenylphosphonates and -carboxylates
13:20–13:35
 Burgart Ya.V., Pryadeina M.V., Khudina O.G., Saloutin V.I.,
Chupakhin O.N. (Russia)
Synthesis of fluoroalkyl-containing pyrimidines
13:35–13:50
 Eremkin A.V., Mol'kov S.N., Ershov O.V. (Russia)
Hydrolysis of cyano groups in 2-halo-6-hydroxy-5,5-dialkyl-
5,6-dihydropyridine-3,4,4(1H)-tricarbonitriles
13:50–14:05
 Gidaspov A.A. (Russia)
bis-Trinitromethylation of 2,4,6-trichloro-1,3,5-triazine
 
14:05–15:00 Lunch
 
 
Oral Presentations

Session Chairpersons: Prof. R. Kostyanovsky, Prof. A. Mikhal'chuk

15:00–15:15
 Gornostaev L.M., Arnold E.V., Beresnev V.A., Dolgushina L.V.,
Lavrikova T.I., Sokolova M.S. (Russia)
Anthraquinone derivatives condensed with pyrrole and triazole rings: Synthesis and properties
15:15–15:30
 Shikhaliev Kh.S., Kryl'skii D.V., Falaleev A.V., Kovygin Yu.A.,
Potapov A.Yu. (Russia)
Construction of heterocyclic systems from guanidines and carbonyls
15:30–15:45
 Gulyakevich O.V., Mikhal'chuk A.L. (Belarus)
Construction of azinone framework by [3+3]-cyclocondensation of
b-enaminones with b-ketoesters
15:45–16:00
 Zobov V.V., Semenov V.E., Kataev V.E., Akamsin V.D., Reznik V.S. (Russia)
Tetraalkylammonium derivatives of uracil and their macrocyclic analogs as potential neuromuscular transmission modulators
16:00–16:15
 Kalinin V.N., Shishkov I.V., Moiseev S.K., Shults E.E.,
Tolstikov G.A. (Russia)
Synthesis of new dienes and trienes of the morphinan series
16:15–16:30
 Kofanov E.R., Sosnina V.V. (Russia)
Multifunctional heterocyclic compounds from nitriles of aromatic
carboxylic acids
16:30–16:45
 Kravchenko A.N., Sigachev A.S., Chikunov I.E., Lozhkin B.V., Baranov V.V., Gazieva G.A., Trunova N.S., Lysenko K.A., Belyakov P.A.,
Makhova N.N. (Russia)
New horizons in a-ureidoalkylation

16:45–17:00 Coffee Break


Oral Presentations

Session Chairpersons: Prof. A. Shestopalov, Prof. Kh. Shikhaliev

17:00–17:15
 Levkovskaya G.G., Bozhenkov G.V., Savosik V.A., Mirskova A.N. (Russia)
Derivatives of 4- and 5-halopyrazoles: Targeted synthesis, structure, and properties
17:15–17:30
 Levinson F.S., Ermolaeva E.A., Efimov S.I., Evgen'ev M.I., Varganov R.V., Vasyutina E.A., Shakirova I.M. (Russia)
4,6-Dichloro-5,7-dinitro- and 4-methoxy-6-chloro-5,7-dinitrobenzofurazans as new two-position electrophiles
17:30–17:45
 Levkovich M.G. (Uzbekistan)
Electric charge on atoms and physicochemical properties of alkaloids
17:45–18:00
 Mareev A.V., Pavlov D.V., Khatashkeev A.V., Medvedeva A.S., Afonin A.V., Ushakov I.A. (Russia)
Cascade assembling of polyfunctional 1,2-dihydropyridine and related compounds from 3-trimethylsilyl-2-propynal and 2-aminopyridine under microwave activation
18:00–18:15
 Musienko Î.À., Dybenko À.G., Kartsev V.G. (Ukraine)
Benzo analogs of cuscutamine and canthine
18:15–18:35
 Nekrasov D.D., Obukhova A.S. (Russia)
2-Amino-substituted 6-aryl-1,3-oxazin-4-ones: Synthesis and biological activity
 

9:00–19:00  Poster Session 3 (poster nos. 151–223) (The Lobby of the Assembly Hall,
the Big Reception-Room)
 
Poster nos.
Poster Details

151

 Ostras' K.S., Gorobets N.Yu., Lukinova E.V., Desenko S.M.
Microwave-assisted three-component synthesis of 4,5,6,7-tetrahydro[1,2,4]­triazolo[1,5-a]pyrimidines

152

 Ostroglyadov E.S., Vasil'eva O.S., Zobacheva M.M., Berestovitskaya V.M.
Potentially bioactive spiropyrrolidones

153

 Pokhodylo N.T., Matiichuk V.S., Tsyalkovskii V.M., Obushak M.D.
Transformations of 5-benzyl-2-imino-4-thiazolidinones

154

 Polygalova N.N., Mikhailovskii A.G., Limanskii E.S., Syropyatov B.Ya., Ismailova N.G., Vakhrin M.I.
New isoquinolines with cardiovascular activity

155

 Popil'nichenko S.V., Chernega A.N., Brovarets V.S.
Reaction of 2-acylamino-3-chloroacrylonitriles with benzamidine and
2-aminonopyridine

156

 Potikha L.Ì., Kovtunenko V.À., Tarasevich À.V.
Oxidation reactions during thermal rearrangement of
7,12-dihydro-5Í-isoquino[2,3-à]quinazolin-5-one

157

 Pryadeina M.V., Burgart Ya.V., Saloutin V.I.
Synthesis of substituted and condensed azoles

158

 Rakhimov Sh.B., Alimova M., Vinogradova V.I.
Reaction of ytosine with benzaldehydes

159

 Ravina I., Zicane D., Tetere Z.
1-Acyl-5-amino-4-carbethoxypyrazoles from monohydrazides
of cyclohexenedicarboxylic acids

160

 Rikkel M.A., Zobov V.V.
Pharmacological properties of uracil-containing haloperidol analog

161

 Romanov D.V., Moiseev S.V., Lyamin A.I., Ivanovskaya N.P., Osin N.S., Semochkin A.V., Vasil'ev N.V.
Fluorinated heterocyclic chelates for immunofluorescent analysis

162

 Romashov K.V., Trostina A.V., Levov A.N., Varlamov A.V.
7-Acylaminopyrido[1,2-a]benzimidazoles: Synthesis and transformations

163

 Rubinov D.B., Rubinova I.L., Zheldakova Ò.À.
3-Acyl-2,4(1Í,3Í)-pyridinediones and their exo- and endo-enamino derivatives

164

 Rudenko R.V., Desenko S.M., Musatov V.I.
Arylidene derivatives of 5-acetylbarbituric and dehydroacetic acids in reaction with aminoazoles

165

 Rusinov G.L., Grebenkin K.F., Vorob'eva M.A., Fedorova O.V.,
Chupakhin O.N.
Molecular design of mycobacteria enzyme inhibitors

166

 Saifina D.F., Mamedov V.A., Berdnikov E.A.
Selenazolo[3,4-a]quinoxalin-2(1Í)-ones

167

 Sakhno Y.I., Chebanov V.A., Desenko S.M., Shishkina S.V., Lukinova E.V., Shishkin O.V.
Three-component reaction of phenylpyruvic acid with aminoazoles and aromatic aldehydes

168

 Santos J.L., Yamasaki P.R., Higuchi C.T., Leite C.Q.F., Chung M.C.
Phthalimide hybrid compounds: Design, preparation, and biological activity against Mycobacterium sp.

169

 Saprykina V.A., Vinogradova V.I., Ambartsumova R.F., Sultankulov À., Ibragimov Ò.F., Shakhidoyatov Kh.M.
Cytisines containing N,S-heterocyclic moieties

170

 Satysheva A.G., Shevchenko M.A., Tsupak E.B.
Synthesis of 1-methyl-2-phenylpyrrolo[3,4-c]pyrazol-3-one

171

 Sennikova Å.V., Korshunov Î.Y., Bicherov À.V., Borodkin G.S.,
Kharabaev N.N., Garnovskii À.D.
3-Hydroxy-2-(benzimidazolyl)-1-indanones: Synthesis, tautomerism, complexation

172

 Seregin V.V., Kuznetsov V.V., Makhova N.N.
Synthesis of diaziridines in protic media: Kinetics and mechanism

173

 Serov A.B., Kartsev V.G., Aleksandrov Yu.A.
1,3-Dipolar cycloaddition of acrylamides to azamethine ylides

174

 Shchepin V.V., Kirillov N.F., Bayanova O.B., Silaichev P.S.
Synthesis of 3-R-1,1-tetramethylene-2,3,4,4à,5,10b-hexahydro-
1Í-chromeno[3,4-c]pyridine-2,4,5-triones through the Reformatsky reaction

175

 Shelyakin V.V., Kartsev V.G., Yaremenko A.G., Lozinskii M.O.
Tandem reactions for modification of natural compounds

176

 Shikhaliev Kh.S., Gusakova N.V., Shestakov A.S.
Reaction of 4,6-dimethyl-2-pyrimidinylhydrazine with derivatives of
2-ethoxymethylenemalonic acid

177

 Silaichev P.S., Stepanyan Yu.G., Shchepin V.V.
Aryl 4-aryl-5-cyano-1-R-2,6-dioxopiperidine-3-carboxylates: Synthesis and reaction with amines

178

 Silaichev P.S., Stepanyan Yu.G., Shchepin V.V.
Esters and amides of 2-R-1,3,4-trioxo-2,3-dihydro-1Í,9bÍ-5-oxa-
2-aza-cyclopenta[2,3]cyclopropa[1,2-a]naphthalene-9ñ-carboxylic acids

179

 Silaichev P.S., Stepanyan Yu.G., Shchepin V.V.
3-Substituted alkyl 6-aryl-2,4-dioxo-5-cyano-3-aza-bicyclo[3,1,0]hexane-
1-carboxylates: Synthesis and reaction with amines

180

 Silaichev P.S., Stepanyan Yu.G., Shchepin V.V.
5-Alkyl-6-aryl-3-R-2,4-dioxo-1-cyano-3-aza-bicyclo[3,1,0]hexanes

181

 Slabko O.Yu., Kachanov A.V., Kaminskii V.A.
New electrophilic reactions of tetrahydropyrido[1,2-a]benzimidazoles

182

 Slivchuk S.R., Rusanov E.B., Brovarets V.S.
A convenient approach to 7-substituted 3-arylsulfonylpyrazolo-
[1,5-a]pyrimidines

183

 Smolyar N.N., Yutilov Yu.M., Gres'ko S.V.
4-Amino-6(hetaryl)pyridazin-3-ones:
Synthesis and cardiovascular activity

184

 Sokolova M.S., Tereshchuk S.P., Gornostaev L.M.
Transformations of 1-acylamino-9,10-anthraquinone and 2-acylamino-
1,4-naphthoquinones

185

 Sorotskaya L.N., Nevolina T.A., Krapivin G.D.
Hydroxamic acids based on 5-R-furfurylidene-5(4H)-oxazolones:
Synthesis and some reactions

186

 Strakova I., Strakovs A., Petrova M., Belyakov S.
Nitrogen-containing 3,4-heteroannelated and 3-hetaryl-substituted coumarins

187

 Sukach V.A., Bol'but A.V., Vovk M.V.
New polyfunctional 3,4-dihydropyrimidin-2(1Í)-ones

188

 Sukhotin A.V., Kartsev V.G.
Substituted 2,3,4,5-tetrahydro-1H-1,5-benzodiazepin-2-ones

189

 Sukhotin A.V., Kartsev V.G., Aleksandrov Yu.A.
Amino acids bearing a tetrahydropyrrole moiety

190

 Takibaeva À.Ò., Ibraev Ì.K., Kîzhina Zh.Ì., Gazaliev À.Ì.,
Nurkenov Î.À., Kazerbaeva B.D.
Synthesis of 3-(1-p-nitrophenylethanol-2-yl)oxazolidine-2-thione

191

 Tarabara I.N., Bondarenko Ya.S., Kas'yan L.I.
(9-Aryl-3,5-dioxo-4,9-diazatricyclo[5,3,1,08,10,02,6]undecan-4-yl)carboxylic acids: Synthesis and properties

192

 Teterina N.M., Makhova T.V., Samartseva N.N., Yunnikova L.P., Makhmudov R.R., Bilevich I.O.
N-Arylmethylanilines containing N,O,S-heterocyclic moieties: Synthesis
and antimicrobial activity

193

 Tkachenko Yu.N., Tsupak E.B.
Purino[8',7':2,3]imidazo[5,1-a]isoquinoline-10,12(9H,11H)-diones: Synthesis and reactivity

194

 Tkachuk T.M., Pivovarenko V.G.
Azaheterocycles based on flavonoid glycosides

195

 Tolkunov S.V., Kibal'nyi À.V., Kryuchkov Ì.À., Afonin À.À., Dulenko V.I.
a-3-Chloropropylpyrilium salts in synthesis
of N-containing heterocycles

196

 Tolkunov V.S., Dulenko V.I.
Synthesis of 5Í-hetero[2,3-e]diazepin-4-ones

197

 Trofimov B.A., Petrova O.V., Ushakov I.A., Sobenina L.N., Mikhaleva A.I.
2-(1-Hydroxy-2,2-dicyanoethenyl)-1-methyl-4,5,6,7-tetrahydroindole: Synthesis and unusual rearrangement

198

 Trostina A.V., Borisova T.N., Levov A.N., Voskressensky L.G.
Substituted tetrahydroazocino[4,5-b]indoles

199

 Tsupak E.B., Tkachenko Yu.N.
Pyrrolo[3,2-d]pyrimidine-2,4-diones: Nitration and reduction to amines

200

 Turmukhambetov A.Zh.,Burdel'naya E.V., Mukusheva G.K.,
Agedilova Ì.Ò., Kazantsev A.V., Adekenov S.Ì., Shults E.E.
Reaction of alkaloids with tetramethylammonium iodide

201

 Ulomskii E.N., Shestakova T.S., Deev S.L., Rusinov V.L., Chupakhin O.N.
New method for synthesis of Lamotridgine and other 3,5-diamino-
1,2,4-triazine derivatives

202

 Usol'tseva N.V., Bykova V.V., Kudrik E.V., Anan'eva G.A.,
Zharnikova N.V., Shishkin V.N.
Induction of mesomorphic state in non-mesomorphic porphyrazine derivatives

203

 Vasil'ev N.V., Romanov D.V., Truskanova T.D., Bazhenov À.À.,
Zatonskii G.V.
New cycloaddition reactions of 2,5-bis(perfluoroalkyl)-1,3,4-oxadiazoles

204

 Vdovina S.V., Mamedov V.A., Mustakimova L.V., Gubaidullin A.T.,
Saifina A.F., Litvinov I.A., Reznik V.S.
Chelate compounds containing 3,4-dihydropyrimidin-2(1Í)-îne moieties

205

 Velikorodov A.V., Imasheva N.M.
New carbamate derivatives of 1,4-benzoxazine

206

 Velikorodov À.V., Kovalev V.B., Borisov A.M., Kamanina N.A.
N,N'-Dimethoxycarbonyl-p-benzoquinonediimine in synthesis of carbamate derivatives of indole through the Nenitzescu reaction

207

 Velikorodov À.V., Kovalev V.B., Nagornaya Yu.V., Timchenko Ì.V.
1,3-Dipolar cycloaddition of arenecarbonitrile N-oxides to Ñ-nitroso derivatives of N-arylcarbamates

208

 Vikrishchuk N.I., Suvorova L.Yu., Popov L.D., Vikrishchuk A.D.
Arylvinyl- and hetarylvinyl-substituted 1,2,4-triazoles: Synthesis and alkylation

209

 Vinogradova V.I., Zhurakulov Sh.N., Bobobekova D., Alimova M., Rakhimov Sh.B.
Derivatives of 1-phenyl-1,2,3,4,-tetrahydroisoquinoline

210

 Vishnevskii Yu.V., Vilkov L.V., Ivanov A.A., Kuznetsov V.V.,
Makhova N.N.
Equilibrium geometry of N-chlorosuccinimide

211

 Vydzhak R.N., Panchishin S.Ya., Kartsev V.G.
Polycyclic derivatives of pyrido[1,2-a]pyrimidine

212

 Vypova N.L., Kazantseva D.S., Rakhimov Sh.B., Vinogradova V.I.
N-benzyl derivatives of cytisine: Hemostatic activity

213

 Yamashkin S.A., Oreshkina E.A., Romanova I.S.
Pyrrolo[2,3-h]quinolines from 2,3-dimethyl- and 1,2,3-trimethyl-
4-aminoindoles

214

 Yamashkin S.A., Zhukova N.V., Romanova I.S.
Reaction of 2,3-dimethyl- and 1,2,3-trimethyl-7-aminoindoles with oxalate

215

 Yaremenko À.G., Shelyakin V.V., Lozinskii Ì.Î.
Ìulticomponent synthesis of new N,S-heterocyclic analogs of steroids

216

 Yudashkin A.V., Golovin E.V.
Thermolysis of C-thienyl- and C-selenophenyltetrazoles

217

 Yutilov Yu.M., Smolyar N.N., Svertilova I.A., Gres'ko C.V., Lomov D.A.
Condensed 6-methylpyridazin-3-ones

218

 Zheldakova Ò.À., Rubinov D.B., Rubinova I.L.
Benzimidazole derivatives from alkoximes of cyclohexane b-triketones

219

 Zhukovskaya Î.N., Anisimova V.À., Spasov À.À., Chernikov Ì.V.,
Yakovlev D.S.
Antiserotonin activity of 2-dialkylaminobenzimidazoles

220

 Zhukovskaya Î.N., Anisimova V.À., Spasov À.À., Kosolapov V.A.,
Chernikov Ì.V., Naumenko L.V.
Biological activity of 2-benzylaminobenzimidazoles

221

 Zicane D., Ravina I., Tetere Z., Petrova M.
3-Acylhexenylamido-1,2-dihydroquinazolin-4(3H)-ones from monohydrazides of cyclohexenedicarboxylic acids

222

 Zorina A.V., Peshkov M.D., Shikhaliev Kh.S.
New heterocyclic systems by recyclizaition of arylmaleimides with
N,N-binucleophiles

223

 Zubenko A.A., Fetisov L.N., Zubenko I.V., Sayapina E.A.
1,2,4-Triazolo[3,4-a]phthalazines: Synthesis and bioactivity


Friday,  June 23, 2006

08:00–09:00 Breakfast


Session I                      Chemistry of synthetic and natural heterocycles
(The Assembly Hall, the Big Reception-Room)


Oral Presentations

Session Chairpersons: Prof. Gy. Hajós, Prof. E. van der Eycken

9:00–9:15
 Volochnyuk D.M., Pushechnikov A.O., Pinchuk A.M.,
Tolmachev A.A. (Ukraine)
Fused 1,5,2-diaza- and 1,5,2-oxazaphosphinines: Synthesis and properties
9:15–9:30
 Ol'shevskaya V.A., Zaitsev A.V., Savchenko A.N., Luzgina V.N., Shtil' A.A., Kalinin V.N. (Russia)
Carboranylporphyrins: Synthesis and bioactivity
9:30–9:45
 Ershov A.Yu., Lagoda I.V., Koshmina N.V., Dobrodumov A.V. (Russia)
Recyclization of isoxazole derivatives
9:45–10:00
 Plaskon' A.S., Ryabukhin S.V., Volochnyuk D.M., Tolmachev A.A. (Ukraine)
3-Formylchromones in recyclization with 1,3-CCN- and
1,3-ÑÑÑ-binucleophiles
10:00–10:15
 Makarenko S.V., Berestovitskaya V.M., Sadikov K.D., Tafeenko V.A., Chernyshev I.V. (Russia)
Potentially bioactive 1,4-benzodiazinones and their heteroanalogs:
Synthesis and structure
10:15–10:30
 Medvedeva A.S., Demina M.M., Novokshonov V.V., Safronova L.P.,
Rulev A.Yu., Pavlov D.V., Mareev A.V., Afonin A.V. (Russia)
Synthesis of azidomethyl-1Í-1,2,3-triazoles
10:30–10:45
 Akhmetova V.R., Nadyrgulova G.R., Khairullina R.R., Khafizova S.R., Kunakova R.V., Dzhemilev U.M. (Russia)
One-pot synthesis of novel N,S-containing heterocycles
10:45–11:00
 Mikhalev O.V., Tarasevich B.N., Fedyanin I.V., Il'ina I.G. (Russia)
Autocomplexes of nitroaryls with heterocycles: Synthesis and characterization

11:00–11:30 Coffee Break (The Banquet Hall, the Big Reception-Room)

11:30–13:30 (Lecture-Room 2, The Big Reception-Room)
Round table
·       Moderator: Actagon AB, Stockholm, Sweden
·       Participants: VIP delegates only (including heads of research centers, CEOs of companies and the mayor of the Chernogolovka Research Center)
·       "Prospects for the development of international projects in biotechnology: realization and investment algorithms"


Session I                      Chemistry of synthetic and natural heterocycles
(Session For Russian and CIS Delegates. Working language is Russian)
(The Assembly Hall, the Big Reception-Room)


Oral Presentations

Session Chairpersons: Prof. A. Nemes, Prof. G. Danagulyan

11:30–11:45
 Popkov S.V., Kovalenko L.V. (Russia)
1-Azolylmethyl-6-benzylidene-2-alkoxy-2-methyl- and
2,2-dimethylcyclohexanols: Synthesis and bioactivity
11:45–12:00
 Przheval'skii N.M. (Russia)
Heterohexadiens in synthesis of heterocycles
12:00–12:15
 Samsoniya Sh.A., Trapaidze M.V., Gogrichiani E.O., Katsadze E.A., Maisuradze J.P., Dzhaparidze K.G. (Georgia)
Some spiro derivatives of indole and condensed bis-indoles
12:15–12:30
 Semenov V.E., Nikolaev A.E., Giniyatullin R.Kh., Lodochnikova O.A., Voloshina A.D., Galiullina L.F., Latypov Sh.K., Reznik V.S. (Russia)
Pyrimidinophanes with nitrogen atoms in bridging groups:
Synthesis and properties
12:30–12:45
 Isak A.D., Pogorelova I.P., Tyupalo N.F., Isak V.A. (Ukraine)
Pyrimidine sulfone amides and their derivatives: Synthesis and biological activity
12:45–13:00
 Sirakanyan S.N., Kartsev V.G., Paronikyan E.G., Noravyan A.S. (Armenia)
Derivatives of 2,7-naphthyridine: Synthesis, transformations, and bioactivity
13:00–13:15
 Shestakov A.S., Gusakova N.V., Shikhaliev Kh.S. (Russia)
Cyanamides and their derivatives in reactions of heterocyclyzation
13:15–13:30
 Paronikyan E.G., Noravyan A.S., Hakobyan Sh.F. (Armenia)
New condensed thieno[3,2-d]pyrimidines and thieno[3,2-d]-1,2,3-triazines: Synthesis and bioactivity
13:30–13:45
 Kovalenko S.N., Silin À.V., Savchenko Ò.I. (Ukraine)
Synthesis and reactivity of pyrazolo[4,3-c]quinolines


14:00–16:00 Closing Ceremony and Champagne Party
16:00  Departure