PROGRAM
of the Conference
 
III International Conference on the Chemistry and Biological Activity
of Nitrogen-Containing Heterocycles

June 2023 2006
(Chernogolovka Research Center, Moscow Region, Russia)
 

 
Monday, June 19, 2006

16:0021:00 Registration
(The Hotel of the Chernogolovka Research Center)

Registration of participants of the conference will be held in the Lobby of the Hotel of the Chernogolovka Research Center.

All participants of the conference should have passports.


Tuesday, June 20, 2006

08:00 Registration (The Foyer of the Conference Hall, the House of Scientists)
 
08:30 Breakfast
 
09:00 Opening Ceremony (The Conference Hall, the House of Scientists)
Opening Keynote Address by Prof. Victor G. Kartsev, Chairman of Organizing committee,
Chairman of "Scientific Partnership" Foundation
 
Greetings by honorary delegates of the conference
 

09:30 Presentation ceremony of the Medal "In memory of Professor A.N. Kost"
and the International ScientificPartnership Foundation's awards

 
Scientific Program


Session I Chemistry of synthetic and natural heterocycles


Keynote Lectures

Session Chairpersons: Prof. J. Bergman, Prof. S. Abu-Orabi 

10:3011:00
Mąkosza M. (Poland)
Synthesis of indoles via nucleophilic substitution of hydrogen in nitroarenes
11:0011:40
Van der Plas H.C. (The Netherlands)
The ring transformation as methodology for the synthesis of azaheterocycles

 
11:4012:10 Coffee Break (The Lobby of the Conference Hall, the House of Scientists)


Plenary Lectures

Session Chairpersons: Prof. Henk C. van der Plas, Prof. U. Jordis

12:1012:35
Bergman J., Stensland B. (Sweden)
Novel syntheses of indoles and related heterocycles
12:3513:00
Kartsev V.G. (Russia)
New horizons for use of T-reactions in the synthesis of heterocycles
13:0013:25
Preobrazhenskaya M.N. (Russia)
Chemistry and biology of ascorbigen
13:2513:50
Vasilevsky S.F., Balova I.A. (Russia)
New one-pot synthesis and heterocyclization of vic-functionalized aryl(hetaryl)alkadiynes-1,3
 

14:0015:50 Lunch (Restaurant)
 

Session I Chemistry of synthetic and natural heterocycles 


Plenary Lectures

Session Chairpersons: Prof. M. Mąkosza, Prof. M. Preobrazhenskaya
 
16:0016:25
Fišera L. (Slovak Republic)
Control of regio- and stereoselectivity in nitrone cycloadditions and their utilization in synthesis
16:2516:50
Jordis U. (Austria)
How to use software and integrate databases in the daily practice of heterocyclic chemist
16:5017:15
Hajós Gy. (Hungary)
Zwitter-ionic heterocycles: A pool of novel polyfused ring systems
17:1517:40
Zefirov N.S. (Russia)
Organic chemistry and mathematics: Design and modeling
17:4018:05
Dondoni A., Massi A. (Italy)
Multicomponent synthetic approach to reengineered N-heterocycle pharmacophores by glycoside decoration


Oral Presentations

Session Chairpersons: Prof. L. Fišera, Prof. A. Dondoni

18:0518:25
Nosova E.V., Lipunova G.N., Laeva A.A., Charushin V.N. (Russia)
Fluorinated 2-substituted [1,3]benzothiazinones: Synthesis and properties
18:2518:45
Danagulyan G.G. (Armenia)
KostSagitullin rearrangement with amine exchange and concurrent recyclization of pyrimidinium salts
18:4519:00
Aripova S.F., Zhalolov I.Zh., Levkovich M.G., Tashkhodzhaev B.,
Khuzhaev V.U., Mirzaev Yu.R.
(Uzbekistan)
New alkaloids from Arundo donax L. for medicinal applications
 
 
14:0015:50 Poster Session 1 (poster nos. 175) (The Lobby of the Assembly Hall,
the Big Reception-Room)
 
Poster nos.
Poster Details

1

Aboskalova N.I., Smirnova N.N., Skobeleva A.V., Berestovitskaya V.M.
Synthesis of substituted pyrazoles and isoxazoles from gem-acylnitroethenes

2

Abramov I.G., Voron'ko M.N., Sapegin A.V., Zeifman A.A., Bukhreev P.B., Plakhtinskii V.V.
Phthalonitriles condensed with cycloaliphatic diamines: Synthesis and functionalization

3

Afon'kin A.A., Kostrikin M.L., Shumeiko A.E., Popov A.F.
6,7-Dimethoxy-1-methyldihydroisoquinoline enamines in reactions of
1,2-cycloaddition

4

Agedilova .., Turmukhambetov A.Zh., Kazantsev A.V., Adekenov S.M.
Chemical transformations of vasicinone

5

Akhmedzhanova V.I.
Alkaloids of Haplophyllum perforatum

6

Akhrem A.A., Baranovskii A.V., Gulyakevich O.V., Mikhal'chuk A.L.
Azangular heterocycles: Structure and molecular dynamics as studied
by high-resolution NMR

7

Akhrem A.A., Dubovskii V.L., Gulyakevich O.V., Mikhal'chuk A.L., Tikhomirov S.A., Tolstorozhev G.B.
Absorption/emission properties of 3,4-dihydroisoquinolines: Solvation and acid-base interaction with environment

8

Akhrem A.A., Govorova A.A., Gulyakevich O.V., Lyakhov A.S.,
Mikhal'chuk A.L., Skornyakov I.V., Tolstorozhev G.B.

Intermolecular interactions of immuno-active azasteroids by IR spectroscopy and XRD

9

Akhrem A.A., Gulyakevich O.V., Govorova A.A., Kurman P.V.,
Lyakhov A.S., Mikhal'chuk A.L.

3-Acetyl-4-methylpyrido[2,1-a]isoquinoline-2-ones.
[2+4]-Cyclocondensation of 3,4-dihydroisoquinolines with triacetylmethane

10

Akopyan Sh.F.
Pyrimidine derivatives in synthesis of condensed triazolo-, tetrazolo-, and imidazolopyrimidines

11

Aksenov A.V., Trifonov V.V., Goncharov V.I.
2,3'-Biquinoline derivatives by Vilsmeier reaction

12

Amiranashvili L.Sh., Merlani M.I.
17-Aza-16,17a-D-homoandrost-2-ene from tigogenine

13

Andreev G.N., Shults E.E., Tolstikov G.A.
Synthesis of 5,5-cyclofused barbituric acids

14

Andriyankova L.V., Mal'kina A.G., Nikitina L.P., Trofimov B.A.
Functionalized polyconjugated 1,4-dihydropyridines from pyridine and phenylcyanoacetylene

15

Angenot L., Akhmedzhanova V.I., Akhmedkhodzhaeva Kh.S.,
Nazrullaev S.S.

Biological activity of alkaloids from plants of the Haplophyllum genus

16

Anisimova N.A., Ladygin V.V., Berestovitskaya V.M.
Synthesis of functionalized carbazoles

17

Anisimova V.A., Tolpygin I.E., Askalepova O.I.
Interaction of 2,9-disubstituted imidazo[1,2-a]benzimidazoles
with tetracyanoethylene

18

Anisimova V.A., Tolpygin I.E., Askalepova O.I.
Synthesis of 2,3-dihydroimidazo- and 2,3,4,10-tetrahydropyrimido-
[1,2-a]benzimidazolyl-N-acetic acids and their derivatives

19

Arsen'eva M.Yu., Arsen'ev V.G., Minkin V.I.
New derivatives of furo[3',4':3,4]cyclohepta[d]imidazoles

20

Babakova M.N., Vlaskina N.M., Suzdalev K.F., Mezheritskii V.V.,
Kartsev V.G.

-Reactions in synthesis of condensed a-carbolines

21

Bakbardina O.V., Pukhnyarskaya I.Yu., Fazylov S.D., Gazaliev A.M.
Potassium b-aminoethylxanthogenates from alkaloids

22

Bakbardina O.V., Rakhimzhanova N.Zh., Gazaliev A.M., Fazylov S.D.
New carbamoyloxamidinesfrom anabasine and cytosine

23

Bakharev V.V., Gidaspov A.A.
Alkylation of 5-trinitromethyltetrazolo[1,5-a]-1,3,5-triazine salts

24

Bannikova Yu.N., Khalturina V.V., Sedegova E.A., Maslivets .N.
Heterocyclization of 2,3-dihydro-2,3-pyrrolediones under the action
of binucleophiles

25

Bauman V.T., Shults E.E., Tolstikov G.A.
Synthesis of C(1)-substituted pyrrolidinothebaines

26

Begunov R.S., Ryzvanovich G.A., Nozdracheva O.I.
Condensed pyridines containing a central nitrogen atom

27

Belov E.Yu., Tomachinskii S.N., Dybenko A.G.
Amino-acid modification of spinaceamine

28

Belyuga A.G., Balya A.G., Brovarets V.S.
Recyclization of 4-acylamino-5-aryl-2-phenacylthio-1,3-oxazoles upon heating in polyphosphorous acid

29

Biitseva .V., Gordienko .V., Kornilov .Yu., Sukach V.., Vovk .V.
Regioselective cyclocondensation of 1-arylimino-1-isoindole-3-amines with a-chlorobenzyl isocyanates

30

Bilokin' M.D., Pivovarenko O.V., Yushchenko D.A., Duportail G., Mely Y., Pivovarenko V.G.
New derivatives of 3-hydroxyquinolone: Dyes displaying two-band fluorescence

31

Boldashevskii A.V., Ibraev M.K., Fazylov S.D., Gazaliev A.M., Nukhuly A.
bis-Thioethers from alkaloids and their analogs

32

Bondarenko S.P., Frasinyuk M.S., Khilya V.P.
Heteroanalogs of isoflavone in reaction with hydroxylamine

33

Borisova Yu.Yu., Mironov V.F., Burnaeva L.A., Amerkhanova N.K., Konovalova I.V.
Nitrogen-containing heterocycles from phosphorylated derivatives of hydroxynicotinic acid

34

Borisova Yu.Yu., Mironov V.F., Burnaeva L.A., Amerkhanova N.K., Konovalova I.V.
Reactions of 2-R-benzo[d]-1,3,2-oxazaphosphorin-6-ones with compounds containing activated multiple bonds

35

Borovik V.P., Shkurko O.P.
2-Thio derivatives of 4-phenyl-9H-pyrimido[4,5-b]indole

36

Bulychev Yu.N., Bakharev V.V., Gidaspov A.A.
Cytotoxic activity of 2-R1-4-R2-6-trinitromethyl-1,3,5-triazines

37

Bulychev Yu.N., Bakharev V.V., Gidaspov A.A.
Cytotoxic activity of 3,4-di(2'-R1-4'-R2-1,3,5-triazin-6'-yl)-1,2,5-oxadiazole-N-oxides

38

Butov G.M., Parshin G.U., Panyushkina O.A., Mokhov V.M.
New methods for synthesis of (1-adamantyl)azoles

39

Buzykin B.I., Kovalenko V.I., Ginzburg B.M., Nurgatin V.V.
1,4,5,8,9,10-Hexaazaperhydrodiethano[4,9][8,10]anthracene

40

Bykov E.E., Lakatosh S.A., Preobrazhenskaya M.N.
Reaction of bisindolylmaleimides with protic acids: Quantum-chemical study

41

Bykova V.V., Usol'tseva N.V., Anan'eva G.A., Znoiko S.A., Maizlish V.E., Shaposhnikov G.P.
Copper phthalocyanines containing benzotriazole fragments: Synthesis and mesomorphism

42

Chesnyuk A.A., Mikhailichenko S.N., Zaplishnyi V.N., Neshchadim N.N., Konyushkin L.D.
A new conjugated heterocyclic system, 2-(1-pyrrolyl)-4,6-disubstituted 1,3,5-triazine

43

Chikvaidze I.Sh., Samsoniya Sh.A., Targamadze N.L., Samsonia N.Sh., Kalatozishvili A.Z., Narimanidze N.O., Barbakadze N.N.
New polycyclic heterocycles containing indole and pyridazine moieties

44

Chukhajian E.O., Nalbandyan M.K., Gevorkyan H.R., Khachatryan ..
Intramolecular recyclization of isoindolinium salts and their condensed analogs

45

Churikov D.G., Kulinkovich O.G.
Transformation of carboxylic esters into 5-substituted isoxazoles

46

Dabaeva W.W., Bagdasaryan M.P., Noravyan A.S.
1-Amino-3H-6,6,7-trimethylpyrazolo[3,4-b]-
5,6,7,8-tetrahydro[1,6]naphthyridine dihydrochloride: Synthesis and
anti-monoaminooxydase effect

47

Danagulyan G.G., Boyakhchyan A.P., Sahakyan L.G., Danagulyan A.G.
Synthesis and recyclization of some azolo[1,5-a]pyrimidines

48

Danagulyan G.G., Tadevosyan D.A., Hakobyan V.P., Balasanyan M.G., Ashrafyan K.B.
Synthesis and cerebrovascular activity of some pyrazolo[1,5-a]pyrimidines

49

Deev S.L., Rusinov V.L., Ulomskii E.N., Shestakova T.S., Chupakhin O.N., Kukhanova M.K., Khandazhinskaya A.L., Shirokova E.A.
Abnormal nucleosides from 1,2,4-triazolo[5,1-c][1,2,4]triazin-7-ones

50

Demidchuk B.A., Brovarets V.S., Chernega A.N.
Cyclocondensation of 1-aryl-1,3,4,4-tetrachloro-2-aza-1,3-butadienes with
2-aminobenzimidazole and its homologs

51

Detistov A.S., Zaremba O.V., Kovalenko S.N.
Combinatorial library of 5-(5-methyl-1H-1,2,3-triazol-4-yl)-
1,2,4-oxadiazoles

52

Dimukhametov M.N., Abdrakhmanova L.M., Mironov V.F., Ivkova G.A., Zagidullina E.R., Musin R.Z.
5,7-Dioxa-1-aza-6-phospha-benzo[3,4]bicyclo[4,3,1]decane-2,6-diones through intramolecular cycle expansion in
2-benzylideneminoethyl(phenyl) salicyl phosphites

53

Dimukhametov M.N., Mironov V.F., Abdrakhmanova L.., Musin R.Z.
Reaction of iminophenols with chlorophosphites as a new route to
N,P-containing mcroheterocycles

54

Dmitriev A.S., Abaev V.T., Pilipenko A.S., Podelyakin S.A., Gavrilov .., Butin .V.
Amides of o-carboxybenzylfuran in synthesis of isoquinolone derivatives

55

Dmitrieva I.G., Dyadyuchenko L.V., Kaigorodova E.A.
4,6-Dimethyl-5-R-3-cyanopyridyl-2-sulfonyl chlorides

56

Dotsenko V.V., Krivokolysko S.G., Litvinov V.P.
New derivatives of pyridin-4(1H)-one from diketene and cyanothioacetamide

57

Dubovik I.P., Garazd .., Vinogradova V.I., Khilya V.P.
Modification of cytisine with coumarinyloxyacetic acids

58

Dyachenko V.D.
cross-Recyclizationof4-alkyl(aryl, heteryl)-2,6-diamino-3,5-dicyano-
4H-thio(seleno)pyrans

59

Dybenko A.G., Yazlovitskii A.V., Patrikei S.Yu.
New peptoids bearing a heterocyclic fragment

60

Dzhavakhishvili S.G., Gorobets N.Yu., Paponov B.V., Desenko S.M.
Transformations of Gewald amides in their reactions with aldehydes

61

Egamov D.I., Yakubov U.M., Shakhidoyatov Kh.M.
Reaction of quinazolone thioimidium salts with aromatic amines

62

Elmuradov B.Zh., Shakhidoyatov Kh.M.
O-Alkyl derivatives of quinazoline alkaloids

63

Elmuradov B.Zh., Shakhidoyatov Kh.M.
Reaction of α-oxymethylidene-2,3,4,10-tetrahydro-1H-pyrido-
[2,1-b]-quinazolin-10-one with anabasine and cytisine

64

Elmuradov B.Zh., Turdibaev Zh.E., Shakhidoyatov Kh.M.
a-Piperazinylmethylidene derivatives of quinazoline alkaloids

65

Eshmatov A.K., Topchieva T.S., Andreev S.A., Tashmukhamedova .K.
Phenazine derivatives from dibenzo-18-crown-6

66

Fedorova O.V., Zhidovinova M.S., Ovchinnikova I.G, Valova M.S.,
Kharchuk V.G, Rusinov G.L.

New approaches to multicomponent synthesis of azaheterocycles and heterocycle-containing podands

67

Frasinyuk M.S., Khilya V.P.
Aminomethylation of 2-amino-3-(2-benzothiazolyl)chromones

68

Frolov K.., Dotsenko V.V., Krivokolysko S.G., Litvinov V.P.
New tetrahydronicotineamide derivatives

69

Frolov K.., Dotsenko V.V., Krivokolysko S.G., Litvinov V.P.
Reduction of ()-3-aryl-2-(thiazole-2-yl)acrylonitriles with LiAlH4

70

Gabrielyan S.H., Markosyan A.I.
Some transformations of 3-furfuryl-4-oxo-2-thioxo-
1,2,3,4,5,6-hexahydrospiro(benzo[h]quinazoline-5,1'-cyclohexane)

71

Gazaliev A.M., Nurkenov O.A., Adambekova K.A.
Synthesis of 2-(N-diethylthiocarbamoylthio)-3,4-dimethyl-5-phenyl-
1,3,2-oxazphospholanes

72

Gazaliev A.M., Nurkenov O.A., Aynabaev A.A., Bessonov D.V., Ermukhanbetova R.A.
Chemical modification of some N-xylosyl- and N-glycosylamines

73

Gazaliev A.M., Nurkenov O.A., Sultanov A.S., Ibysheva Sh.T.
New oxazolidines from ephedrine alkaloids

74

Gazieva G.A., Lozhkin P.V., Kravchenko A.N.
Reaction of 4,5-dihydroxyimidazolidin-2-ones with sulfamides

75

Gidaspov A.A.
Trinitromethylation of 2,4,6-trichloro-1,3,5-triazine in the presence of water, alcohols, and phenols
 
 
19:2020:30 Welcome Cocktail Party (The Lobby of the Conference Hall, the House of Scientists)
 

Wednesday, June 21, 2006
 

8:30 Breakfast


Session I Chemistry of synthetic and natural heterocycles 

Keynote and Plenary Lectures (The Assembly Hall, the Big Reception-Room)

Session Chairpersons: Prof. H.-J. Knölker, Prof. S. Vasilevsky 

9:009:30
Atta-ur-Rahman, Choudhary M.I. (Pakistan)
Nitrogen-containing heterocycles from natural sources: Isolation, biological studies, and synthesis
9:309:55
Florio S. (Italy)
o-Lithiation: a useful strategy towards heterocycles
9:5510:20
Chupakhin O.N., Rusinov V.L., Charushin V.N. (Russia)
Abnormal nucleosides from isosteres of purine

Oral Presentation
 
10:2010:35
Van der Eycken E. (Belgium)
Microwave irradiation: A 'green tool' in 2(1H)-pyrazinone chemistry

Plenary Lecture 

10:3511:05
will be announced later
 
11:1011:30 CoffeeBreak (The Banquet Hall, the Big Reception-Room)
 
Oral Presentations

Session Chairpersons: Prof. O. Chupakhin, Prof. S. Florio

11:3012:00
Agarwal S., Filali S., Fröhner W., Knöll J., Krahl M.P., Reddy K.R.,
Knölker H.-J. (Germany)
Application of oxidative cyclizations to the synthesis of bioactive
nitrogen-containing heterocycles
12:0012:15
Abu-Orabi S.T. (Jordan)
Utilization of 1,2,3-dipolar cycloaddition reactions of azides toward
the synthesis of 5-membered rings heterocyclic compounds
12:1512:30
Nemes A. (Hungary)
Synthetic studies related to cis- and trans-apovincamine derivatives and metabolites
12:3013:00
Rádl S., Klecán O. (Czech Republic)
New approaches to the synthesis of triptans
13:0013:15
Bölcskei H., Gács-Baitz E., Szántay Cs. Jr., Kalaus Gy.,
Szántay Cs.
(Hungary)
Synthesis of indoloazepines and indoloazocines
13:1513:30
Geronikaki A., Incerti M., Zani F., Vicini P. (Greece)
2-Benzo[d]isothiazolylimino-5-arylidene-4-thiazolidinones: Synthesis and antimicrobial activity
13:3013:45
Shklyaev Yu.V., Glushkov V.A., Stryapunina O.G., Rozhkova Yu.S.,
El'tsov M.A. (Russia)
The synthesis of partially hydrohenization azine and azole: Dihydroisoquinolines, spiropyrrolines, polyhydroindolines

13:4515:15 Lunch (Restaurant)
 

Session I Chemistry of synthetic and natural heterocycles

Oral Presentations
 
Session Chairpersons: Prof. S. Rádl, Prof. A. Geronikaki

15:1515:30
Bazureau J.P., Legeay J.C., Fraga-Dubreuil J., Hakkou H. (France)
Ionic liquid-phase technology: A new tool for combinatorial chemistry. Applications in heterocyclic chemistry mediated by microwave
dielectric heating
15:3015:45
Voskressensky L.G., Vorob'ev I.V., Varlamov A.V. (Russia)
Unusual reactions of tetrahydrobenzo[b][1,6]naphthyridines with activated alkynes
15:4516:00
Korotkikh N.I., Raenko G.F., Kiselev .V., Knishevitsky .V., Shvaika .P., Glinyanaya N.V., Panov I.S., Cowley .H., Jones J.N., Moore J.A. (Ukraine)
Stable carbenes. Insertion into і bonds and reaction with ester function. New cleavage and thermal transformation of 1,2,4-triazol-5-ylidenes
16:0016:15
Stroganova T.A., Vasilin V.K., Krapivin G.D. (Russia)
Amino acids of the thieno[2,3-b]pyridine series in reactions of intramolecular cyclization
16:1516:30
Gorobets N.Yu., Ermolaev C.A., Dzhavakhishvili S.G., Sirko S.N., Chernenko V.N., Desenko S.M. (Ukraine)
2-Dimethylaminomethylene-1,3-cyclohexanedione derivatives in reaction with methylene-active nitriles
16:3016:45
Makhova N.N., Shevtsov A.V., Petukhova V.Yu., Kuznetsov V.V.,
Kislukhin A.A.
(Russia)
Transformation of diaziridine ring under the action of ketenes as a new synthetic approach to nitrogen-containing heterocyclic systems
16:4517:00
Polygalova N.N., Mikhailovskii A.G., Vakhrin M.I. (Russia)
Carbonyl derivatives of condensed isoquinolines: Synthesis and reactivity
 
17:0017:20 Coffee Break
 

Oral Presentations

Session Chairpersons:Prof. J.P. Bazureau, Prof. H. Bölcskei, Prof. L. Voskressensky

17:2017:35
Suzdalev K.F., Babakova M.N., Den'kina S.V, Kartsev V.G. (Russia)
Indoles bearing reactive groups for synthesis of combinatorial libraries
17:3517:50
Vizer S.A., Dedeshko E.H., Erzhanov K.B., Dembitskii V.M. (Kazakhstan)
Synthesis of N-containing heterocycles from a-propargyl-b-dicarbonyls and their O-phosphoryl derivatives
17:5018:05
Lesyk R.B., Zimenkovsky B.S., Atamanyuk D.V. (Ukraine)
Thiopyrano[2,3-d]thiazoles and their derivatives: Synthesis and biological activity
18:0518:20
Kozminykh V.O., Goncharov V.I., Kozminykh E.N., Fiergang S.I. (Russia)
Synthesis of oxoalkylidene(oxocycloalkyl)quinoxalinones


Session II Biological activity of nitrogen-containing heterocycles
(Lecture-Room 2, The Big Reception-Room)

Plenary Lectures
  
Session Chairpersons: Prof. N. Zefirov, Prof. . Saxena, Prof. V. Poroikov

15:0015:25
Zefirov N. (Russia)
The use of QSAR in the search of biologically active compounds
15:2515:50
Poroikov V.V., Filimonov D.A., Gloriozova T.A., Lagunin A.A. (Russia)
Computer-aided prediction of biological activity for nitrogen-containing organic compounds
15:5016:15
Saxena . (India)
Substituted arylpiperazines in rational drug design

Oral Presentations
 
16:1516:30
Mali A., Shelar M., Shelar A. (India)
Antibiotic resistance: A search for new b-lactam antibiotics
16:3016:45
Chung M.C. (Brazil)
Prodrug design: Improving drug activity
16:4517:00
Belous A.R. (USA)
Endogenous indole compounds: biological significance of
5-hydroxytriptamine and its metabolites
 
17:0017:20 Coffee Break

 
Oral Presentations
 
17:2017:35
Granzhan A., Ihmels H., Viola G. (Germany)
Rearrangements in diazoniapentaphenes and DNA-binding properties
of diazoniapolycycles
17:3517:50
Duburs G., Bisenieks E., Krauze A., Plotniece A., Sobolevs A., Tirzitis G., Vigante B. (Latvia)
Dihydropyridine derivatives as biomimetics and bioprotectors
17:5018:05
Veinberg G., Vorona M., Shestakova I., Kanepe I., Lukevics E. (Latvia)
Antitumor 3a-chloro- and 3-alkylideneazetidinone-2 derivatives

 
9:0019:00 Poster Session 2 (poster nos. 76150) (The Lobby of the Assembly Hall,
the Big Reception-Room)
 
Poster nos.
Poster Details

76

Gladkov E.S., Desenko S.M., Sirko S.N.
Three-component cyclocondensation of aminoazoles with cyclic ketosulfones and aldehydes

77

Gorbulenko N.V., Kurdyukova I.V., Turov .V., Khilya V.P.
2-Aminoimidazo[1,5-a]pyrimido[5,4-c]quinolin-10-ol as a new condensed heterocyclic system

78

Gorbulenko N.V., Tkachuk .M., Shokol .V., Semenyuchenko V.V.,
Khilya V.P.

Annelation of oxazine cycle to 3-hetarylchromones through Mannich's reaction

79

Gorichko M.V., Komarov I.V., Patrikei S.Yu.
Conformationally rigid analogs of cyclic a-amino acids

80

Gulyakevich O.V., Mikhal'chuk A.L., Akhrem A.A.
[2+4]-Cyclocondensation of cyclic Schiff bases with b-di-, b,b'-tricarbonyl compounds: Perycyclic heterocyclization of iminium cations with enol anions of b-di-, b,b'-tricarbonyl compounds

81

Gusakova N.V., Shikhaliev Kh.S., Shestakov A.S.
Regioisomeric pyrazoles from 4,6-dimethylpyrimidinyl-2-hydrazine and esters of 3-oxoacids

82

Ibraev .K., Kzhin Zh.., Gzliev .M., Fazylov S.D., Takibaeva A.T.
N-[(5-thioxo-4,5-dihydro-1,3,4-oxa-diazol-2-yl)methyl]benzamides

83

Ibragimov .F., Saprykina V.A., Shakhidoyatov Kh.M.
Condensation of heterocyclic amines with N-methylol lactams

84

Isaikina O.G., Kalinin A.A., Mamedov V.A.
Tiazolo[3,4-a]quinoxaline monopodands from
bis-3-(a-bromoethyl)quinoxalin-2-ones and thiourea

85

Ishchenko V.V., Shablykina O.V., Shablykin O.V., Khilya V.P.
3-Hetarylisocoumarins: Synthesis and transformation into
3-hetarylisoquinolones

86

Ivanov S.P., Nugumanov T.R., Spirikhin L.V., Murinov Yu.I.
4-Methyl-5-hydroxyuric acid from 5-hydroxy-6-methyluracil
in aqueous solution

87

Ivkova G.A., Mironov V.F., Burnaeva L.M., Konovalova I.V.,
Shemetova A.S., Ogurtsova E.V.

2,5-Dioxobenzo[f]-1,4,2-oxazaphosphepines by reaction of 3-alkyliminopyridines with salicylphosphites

88

Kagarlitskii A.D., Balpanov D.S., Krichevskii L.A., Postnikov L.S.
Oxidative ammonolysis of 2-methyl-3-hydroxyquinoxaline

89

Kalinichenko .N., Zhernosek .V., Litvinko N.., Kuchuro S.V.,
Rakhuba G.N.

2',3'-Dideoxycytidine-5'-monophosphate-phosphatidylethanolamine-phosphoramidate: Synthesis and interaction with phospholipase 2

90

Kartsev V.G., Serov A.B., Sukhotin A.V.
New derivatives of couroupitine A (tryptanthrine): Synthesis and transformations

91

Kas'yan L.I., Karpenko D.V., Kas'yan A.O.
Reaction of norbornene sulfonamides with organic peracids

92

Katorov D.V., Illarionova T.A., Rudakov G.F., Zhilin V.F.
Synthesis of heterocyclic geminal nitroazides

93

Khilya O.V., Vintonyak V.V., Volovenko Yu.M.
Reaction of hetarylacetonitriles with heterocyclic 1,3-bielectrophilic halocarbonyls

94

Khudina O.G., Shchegol'kov E.V., Burgart Y.V., Saloutin V.I.
Ringchain transformations of 7-fluoroalkyl-4,7-dihydroazolo[5,1-c]triazines in reaction with hydrazides and thiosemicarbazide

95

Kislukhin ., Shevtsov .V., Kuznetsov V.V., Makhova N.N.
N-acyl- and N,N-bisacylpyrazolidines from 1,5-diazabicyclo[3,1,0]hexanes and acyl chlorides

96

Kolobov A.V., Panfilov S.T., Borisov P.V., Kofanov E.R.
Arylpyridazines: Synthesis, structure, chemical behavior

97

Kol'tsov N.Yu.
Reduction of heterocyclic a-aminonitriles with lithium aluminum hydride

98

Komykhov S.A., Petrova M.G., Borovskoi V.A., Musatov V.I.,
Desenko S.M.

New dihydropyrazolo[1,5‑a]pyrimidine derivatives by three-component condensation of 3-aminopyrazole-4‑arylcarboxamides with carbonyls

99

Kopteva N.I., Stepanova T.V.
Heterocyclization of coumarin-3-carboxylic acid hydrazide

100

Korotkikh N.I., Kiselev .V., Kovalenko A.N., Shvaika O.P., Cowley .H., Jones J.N., Moore J.A.
New routes to synthesis of carbene complexes with alkali and transition metals from heteroaromatic carbenes and their precursors

101

Koshchienko Yu.V.
Synthesis of dihetarylphenylcarbinols involving organometallic compounds

102

Kostenev I.S., Ovcharov M.V., Voskressensky L.G., Varlamov A.V.
Heteroannelated pyridopyrimidines: Synthesis and transformations

103

Kostenko E.S., Kaigorodova E.A., Krapivin G.D.
4-(3-Pyridyl)-1,6-dihydro-6-pyrimidinones

104

Kostrub V.V., Shevchenko M.A., Tsupak E.B.
Pyrimido[d]pyriliuim salts in synthesis of new fused nitrogen-containing heterocycles

105

Kovalenko S.N., Vlasov S.V., Silin A.V., Chernykh V.P.
Reaction of 2-iminocoumarin-3-carboxamides with 2-aminothiobenzamide

106

Krasnov V.P., Levit G.L., Zhdanova E.A., Solieva N.Z., Sadretdinova L.Sh., Chupakhin O.N.
Kinetic resolution of racemic piperidine derivatives

107

Kryl'skii D.V., Shikhaliev Kh.S., Didenko V.V.
Heterocyclic systems from aminopyrazoles and diketones

108

Kryl'skii D.V., Shikhaliev Kh.S., Didenko V.V.
Pyrazolotriazines from aminopyrazoles and -active compounds

109

Krysin M.Yu., Petrov V.V., Muratov D.N.
Indeno[1,2-d]pyrimidines from 2-arylidene-1,3-indandiones and guanidines

110

Kurbatov E.S., Krasnikov V.V., Pavlenko D.A., Mezheritskii V.V.
Rearrangement of pyrano[2,3-d]pyrimidines

111

Kurbatov S.V., Goumont R., Tatarov A.V., Terrier F.
Functionalization of nitrobenzodifuroxan with dienes generated in situ

112

Kutrov G.P., Kovalenko N.V., Cherepakha A.Yu.
Reaction of heterocyclic imidazo bromides with oxidizers

113

Kuznetsov A.Yu., Kholopov U.A., Chapyshev S.V., Nam N.L.
2-Piperidine-substituted 4-aminopyrimidines by reduction of
4-amino-2-pyridylpyrimidines

114

Kuznetsov A.Yu., Kholopov U.A., Chapyshev S.V., Nam N.L.
New 5,6,7,8-tetrahydropyrido[d]pyrimidines

115

Kuznetsov D.V., Neskubo A.A., Andreev S.A., Tashmukhamedova A.K.
2-Amino-5-(-dibenzo-18-crown-6-yl)-thiadiazole

116

Kuznetsov V.V., Makhova N.N.
New stable heterocyclic a-hydroxy-N-chloroalkylamines

117

Kuznetsov V.V., Makhova N.N., Terpigorev A.N.
New method for synthesis of alkyl-substituted diaziridines

118

Ktovskaya S.K., Tzoi ., Charushin V.N.
Fluorinated 3,8-dihydroxyquinolines, analogs of natural antitumor
drug Jeneol

119

Ktovskaya S.K., Zhumabaeva G.., Perova N.., Chupakhin O.N., Charushin V.N.
Tandem SNH(AO) and SNipso(AE) reactions in synthesis of fluorinated 3-amino-1,2,4-benzotriazines

120

Lapteva E.S., Kayukova O.V., Kayukov Ya.S., Ershov O.V.
Substituted 6,6-(2-oxoindol-3,3-ylidene)-3-azabicyclo[3,1,0]hexane-
1,5-dicarbonitriles

121

Levinson F.S., Akimova S.A., Khasanov R.Kh., Sharnin G.P., Efimov S.I., Falyakhov I.F., Ermolaeva E.A., Varganov R.V., Vasyutina E.A.,
Shakirova I.M.

Nitroso- and nitrosonitrohalonitriles in synthesis of 4,6-dichloro- and
4-methoxy-6-chloro-5,7-dinitrofurazan

122

Levinson F.S., Ermolaeva E.A., Kalimullina N.I., Vasyutina E.A.,
Varganov R.V.

4-Aminobenzofurazans containing residua of secondary amines

123

Levinson F.S., Khasanov R.Kh., Sharnin G.P., Gafarov A.N.
Bromonitrobenzofurazans in the Ullmann reaction

124

Levkovich M.G., Proskurina U.G.
Effect of solvent on chemical shifts in 1H NMR spectra of alkaloids

125

Levov N.N., Le Tuan Anh, Komarova A.I., Gimranova G.S., Soldatova S.A., Soldatenkov A.T.
Diarenopiperidinomonoaza-14-crowno-4-phanes: Synthesis and reactions

126

Mamedov V.A., Khafizova E.A., Beschastnova T.N., Rizvanov I.Kh., Berdnikov E.A.
Three-component condensation of pyrid-2-one with bis-(2-chloroethyl)amine hydrochloride as a new method for oxazolidinoethylation

127

Mamedov V.A., Khafizova E.A.
Chelate azolo[a]annelated qunoxalines from phenylhalopyruvates and their structural analogs

128

Marakhovskaya T.G., Shchurova N.A., Tyrkov A.G.
New functionally modified 1,2,3-triazoles based on 5-nitromethyl-
1,2,4-oxadiazoles

129

Markosyan A.I., Dilanyan S.V., Arsenyan F.H., Sukasyan R.S., Garibdzhanyan B.T.
Benzo[h]quinazolines from 1-amino-3-ethyl-3-methyl-2-cyano-
3,4-dihydronaphthalene

130

Maslivets .N., Racheva N.L., Shklyaev Yu.V.
Functionalized spiro-bis-heterocyclic systems

131

Matiichuk V.S., Gorak Yu.I., Lytvyn R.Z., Obushak M.D.
Cyclization of 2-cyl-5-arylfurans

132

Medvedeva S.M., Shikhaliev Kh.S., Solov'ev A.S.
New derivatives of spiro-b-carbolines

133

Mel'chin V.V., Butin A.V.
2-Arylfurans in synthesis of indole derivatives

134

Melekhin E.A., Bardasov I.N., Ershov O.V., Kayukov Ya.S.
2,4-Diamino-7-hydroxy-10-aryl-10-9-oxa-1-azaanthracene-3-carbonitrile

135

Melekhin E.A., Bardasov I.N., Ershov O.V., Kayukov Ya.S.
10-R-5-Aryl-2,4-diamino-8,8-dimethyl-6-oxo-
5,6,7,8,9,10-hexahydrobenzo[b]-1,8-naphthyridine-3-carbonitriles

136

Mel'nikov V.V., Il'ina I.G., Ivanov A.A., Tarasevich B.N.
Autocomplexes of the nitroquinoline series: Synthesis and
spectral investigation

137

Merlani M.I., Amiranashvili L.Sh., Davitishvili M.G.
Ketosteroid hydrazones: Synthesis and bioactivity

138

Mishchenko D.V., Frog E.S., Finegold I.I., Kotel'nikova R.A.,
Bogdanov G.N.

2,4,6-Trimethyl-3-oxypyridine nitrosuccinate as a membranoprotector
at oxidative stress

139

Moiseev S.V., Cherstkov V.F., Vasil'ev N.V.
Synthesis and cycloaddition reactions of polyfluorinated imines and ketones

140

Mol'kov S.N., Eremkin A.V., Ershov O.V.
2-(3-Amino-8-R-1,4-diazaspiro[4,5]dec-3-en-2-ylidene) malonodinitriles

141

Mol'kov S.N., Eremkin A.V., Ershov O.V., Kayukov Yu.S.
5,5,6-Trialkyl-2-halo-6-hydroxy-5,6-dihydro-3,4,4(1)-pyridinetricarbonitriles 5,6-Dialkyl-2-halo-3,4-pyridinedicarbonitriles

142

Mostovaya O.A., Shakirova E.R., Khusainova N.G., Cherkasov R.A.
Reaction of 2H-1,2,3-diazaphosphole with pyrocatechol

143

Mukusheva G.K., Turmukhambetov A.Zh., Kazantsev A.V., Adekenov S.M.
Aminomethylation of glaucine

144

Murav'eva E.A., Chebanov V.A., Musatov V.I., Desenko S.M.
Ultrasound-activated synthesis of 2,4,6-tri- and 2,2,4,6-tetra-substituted 1,2,5,6-tetrahydropyrimidines

145

Musina L.A., Shults E.E., Tolstikov G.A., Adekenov S.M.
Synthesis of substituted indolizines

146

Nagorichna I.V., Garazd .., Garazd Ya.L., Khilya V.P.,
Ogorodniichuk A.S.

Synthesis of linear and angular pyranodihydrobenzoxazines

147

Nekrasov D.D., Obukhova A.S., Kharitonova A.V., Khlbnikova .B.
Stereoisomeric 6-aryl-2-(2-thienyl)-3-(abieta-8,11,13-trien-18-yl)-
1,3-xazin-4-nes

148

Nevolina T.A., Shevlyakov M.V., Stroganova T.A.
Amines of the furan series in synthesis of nitrogen-containing heterocycles

149

Nurmagambetov Zh.S., Turmukhambetov A.Zh., Serperov K.S.,
Kazantsev A.V., Adekenov S.M.

Halogenation of stachydrine

150

Oganisyan Art.Sh., Oganisyan A.Sh., Noravyan A.S.
4,7,7-Substituted pyrano[4',3':4,5]thienoimidazo[1,2-a]pyrimidine-5-diones
 
20:00 Banquet
 
 
Thursday, June 22, 2006
(For Foreign Delegates)

08:00
09:00 Breakfast
9:0014:00 Social events for foreign guests (sightseeing tour of Moscow, the Kremlin, a visit to the Cathedral of Christ-the-Savior, entertainment program)
14:0015:00 Lunch
15:0020:00 Cultural program continued
 
21:00 Snacks & wine party
 
 
Thursday, June 22, 2006
(Session For Russian and CIS Delegates. Working language is Russian)
(The Assembly Hall, the Big Reception-Room)
 
08:0009:00 Breakfast
 

Session I Chemistry of synthetic and natural heterocycles
 
Plenary Lectures 

Session Chairpersons: Prof. Yu. Shklyaev, Prof. L. Gornostaev

9:009:25
Tolstikov G.A. (Russia)
Synthetic transformation of morphinane and diterpene alkaloids
9:259:50
Granik V.G. (Russia)
Biotransformations of heterocyclic nitrogen-containing drugs
9:5010:15
Sagitullina G.P., Sagitullin R.S. (Russia)
Recyclization of pyridinium salts: New horizons
10:1510:40
Akhrem A.A., Gulyakevich O.V., Mikhal'chuk A.L. (Belarus)
[2+4]-Cyclocondensation of monocyclic azomethines with b-di- and
b,b'-tricarbonyl compounds in synthesis of azangular heterocycles
10:4011:05
Kostyanovsky R.G. (Russia)
Nitrogen chirality in heterocyclic chemistry
11:0511:30
Shestopalov A.M., Rodinovskaya L.A., Shestopalov A.A. (Russia)
Recyclization reactions of degenerate carbo- and heterocycles: Practical retrosynthetic approach to new multicomponent methods for synthesis
of N-containing five- and six-membered heterocycles
11:3011:55
Saloutin V.I., Burgart Ya.V., Chupakhin O.N. (Russia)
Design of azaheterocycles based on fluorine-containing 2,4-dioxobutanoates and their derivatives
 
12:0012:20 CoffeeBreak (The Banquet Hall, the Big Reception-Room)
 

Oral Presentations

Session Chairpersons: Prof. G. Tolstikov, Prof. V. Granik

12:2012:35
Drach B.S., Sviripa V.N., Pil'o S.G., Popil'nichenko S.V., Golovchenko A.V., Brovarets V.S. (Ukraine)
Synthesis of functionalized condensed heterocycles from 2-acylamino-
3,3-dichloroacrylonitriles
12:3512:50
Velikorodov .V. (Russia)
Quinones and quinoids in synthesis and modification of indoles
12:5013:05
Adekenov S.. (Kazakhstan)
Nitrogen-containing derivatives of natural sesquiterpene lactones
13:0513:20
Berestovitskaya V.M., Anisimova N.A., Makarova N.G. (Russia)
Synthesis of nitrogen-containing heterocycles from
b-nitroethenylphosphonates and -carboxylates
13:2013:35
Burgart Ya.V., Pryadeina M.V., Khudina O.G., Saloutin V.I.,
Chupakhin O.N.
(Russia)
Synthesis of fluoroalkyl-containing pyrimidines
13:3513:50
Eremkin A.V., Mol'kov S.N., Ershov O.V. (Russia)
Hydrolysis of cyano groups in 2-halo-6-hydroxy-5,5-dialkyl-
5,6-dihydropyridine-3,4,4(1H)-tricarbonitriles
13:5014:05
Gidaspov A.A. (Russia)
bis-Trinitromethylation of 2,4,6-trichloro-1,3,5-triazine
 
14:0515:00 Lunch
 
 
Oral Presentations

Session Chairpersons: Prof. R. Kostyanovsky, Prof. A. Mikhal'chuk

15:0015:15
Gornostaev L.M., Arnold E.V., Beresnev V.A., Dolgushina L.V.,
Lavrikova T.I., Sokolova M.S. (Russia)
Anthraquinone derivatives condensed with pyrrole and triazole rings: Synthesis and properties
15:1515:30
Shikhaliev Kh.S., Kryl'skii D.V., Falaleev A.V., Kovygin Yu.A.,
Potapov A.Yu.
(Russia)
Construction of heterocyclic systems from guanidines and carbonyls
15:3015:45
Gulyakevich O.V., Mikhal'chuk A.L. (Belarus)
Construction of azinone framework by [3+3]-cyclocondensation of
b-enaminones with b-ketoesters
15:4516:00
Zobov V.V., Semenov V.E., Kataev V.E., Akamsin V.D., Reznik V.S. (Russia)
Tetraalkylammonium derivatives of uracil and their macrocyclic analogs as potential neuromuscular transmission modulators
16:0016:15
Kalinin V.N., Shishkov I.V., Moiseev S.K., Shults E.E.,
Tolstikov G.A.
(Russia)
Synthesis of new dienes and trienes of the morphinan series
16:1516:30
Kofanov E.R., Sosnina V.V. (Russia)
Multifunctional heterocyclic compounds from nitriles of aromatic
carboxylic acids
16:3016:45
Kravchenko A.N., Sigachev A.S., Chikunov I.E., Lozhkin B.V., Baranov V.V., Gazieva G.A., Trunova N.S., Lysenko K.A., Belyakov P.A.,
Makhova N.N.
(Russia)
New horizons in a-ureidoalkylation

16:4517:00 Coffee Break


Oral Presentations

Session Chairpersons: Prof. A. Shestopalov, Prof. Kh. Shikhaliev

17:0017:15
Levkovskaya G.G., Bozhenkov G.V., Savosik V.A., Mirskova A.N. (Russia)
Derivatives of 4- and 5-halopyrazoles: Targeted synthesis, structure, and properties
17:1517:30
Levinson F.S., Ermolaeva E.A., Efimov S.I., Evgen'ev M.I., Varganov R.V., Vasyutina E.A., Shakirova I.M. (Russia)
4,6-Dichloro-5,7-dinitro- and 4-methoxy-6-chloro-5,7-dinitrobenzofurazans as new two-position electrophiles
17:3017:45
Levkovich M.G. (Uzbekistan)
Electric charge on atoms and physicochemical properties of alkaloids
17:4518:00
Mareev A.V., Pavlov D.V., Khatashkeev A.V., Medvedeva A.S., Afonin A.V., Ushakov I.A. (Russia)
Cascade assembling of polyfunctional 1,2-dihydropyridine and related compounds from 3-trimethylsilyl-2-propynal and 2-aminopyridine under microwave activation
18:0018:15
Musienko .., Dybenko .G., Kartsev V.G. (Ukraine)
Benzo analogs of cuscutamine and canthine
18:1518:35
Nekrasov D.D., Obukhova A.S. (Russia)
2-Amino-substituted 6-aryl-1,3-oxazin-4-ones: Synthesis and biological activity
 

9:0019:00 Poster Session 3 (poster nos. 151223) (The Lobby of the Assembly Hall,
the Big Reception-Room)
 
Poster nos.
Poster Details

151

Ostras' K.S., Gorobets N.Yu., Lukinova E.V., Desenko S.M.
Microwave-assisted three-component synthesis of 4,5,6,7-tetrahydro[1,2,4]triazolo[1,5-a]pyrimidines

152

Ostroglyadov E.S., Vasil'eva O.S., Zobacheva M.M., Berestovitskaya V.M.
Potentially bioactive spiropyrrolidones

153

Pokhodylo N.T., Matiichuk V.S., Tsyalkovskii V.M., Obushak M.D.
Transformations of 5-benzyl-2-imino-4-thiazolidinones

154

Polygalova N.N., Mikhailovskii A.G., Limanskii E.S., Syropyatov B.Ya., Ismailova N.G., Vakhrin M.I.
New isoquinolines with cardiovascular activity

155

Popil'nichenko S.V., Chernega A.N., Brovarets V.S.
Reaction of 2-acylamino-3-chloroacrylonitriles with benzamidine and
2-aminonopyridine

156

Potikha L.., Kovtunenko V.., Tarasevich .V.
Oxidation reactions during thermal rearrangement of
7,12-dihydro-5-isoquino[2,3-]quinazolin-5-one

157

Pryadeina M.V., Burgart Ya.V., Saloutin V.I.
Synthesis of substituted and condensed azoles

158

Rakhimov Sh.B., Alimova M., Vinogradova V.I.
Reaction of ytosine with benzaldehydes

159

Ravina I., Zicane D., Tetere Z.
1-Acyl-5-amino-4-carbethoxypyrazoles from monohydrazides
of cyclohexenedicarboxylic acids

160

Rikkel M.A., Zobov V.V.
Pharmacological properties of uracil-containing haloperidol analog

161

Romanov D.V., Moiseev S.V., Lyamin A.I., Ivanovskaya N.P., Osin N.S., Semochkin A.V., Vasil'ev N.V.
Fluorinated heterocyclic chelates for immunofluorescent analysis

162

Romashov K.V., Trostina A.V., Levov A.N., Varlamov A.V.
7-Acylaminopyrido[1,2-a]benzimidazoles: Synthesis and transformations

163

Rubinov D.B., Rubinova I.L., Zheldakova ..
3-Acyl-2,4(1,3)-pyridinediones and their exo- and endo-enamino derivatives

164

Rudenko R.V., Desenko S.M., Musatov V.I.
Arylidene derivatives of 5-acetylbarbituric and dehydroacetic acids in reaction with aminoazoles

165

Rusinov G.L., Grebenkin K.F., Vorob'eva M.A., Fedorova O.V.,
Chupakhin O.N.

Molecular design of mycobacteria enzyme inhibitors

166

Saifina D.F., Mamedov V.A., Berdnikov E.A.
Selenazolo[3,4-a]quinoxalin-2(1)-ones

167

Sakhno Y.I., Chebanov V.A., Desenko S.M., Shishkina S.V., Lukinova E.V., Shishkin O.V.
Three-component reaction of phenylpyruvic acid with aminoazoles and aromatic aldehydes

168

Santos J.L., Yamasaki P.R., Higuchi C.T., Leite C.Q.F., Chung M.C.
Phthalimide hybrid compounds: Design, preparation, and biological activity against Mycobacterium sp.

169

Saprykina V.A., Vinogradova V.I., Ambartsumova R.F., Sultankulov ., Ibragimov .F., Shakhidoyatov Kh.M.
Cytisines containing N,S-heterocyclic moieties

170

Satysheva A.G., Shevchenko M.A., Tsupak E.B.
Synthesis of 1-methyl-2-phenylpyrrolo[3,4-c]pyrazol-3-one

171

Sennikova .V., Korshunov .Y., Bicherov .V., Borodkin G.S.,
Kharabaev N.N., Garnovskii .D.

3-Hydroxy-2-(benzimidazolyl)-1-indanones: Synthesis, tautomerism, complexation

172

Seregin V.V., Kuznetsov V.V., Makhova N.N.
Synthesis of diaziridines in protic media: Kinetics and mechanism

173

Serov A.B., Kartsev V.G., Aleksandrov Yu.A.
1,3-Dipolar cycloaddition of acrylamides to azamethine ylides

174

Shchepin V.V., Kirillov N.F., Bayanova O.B., Silaichev P.S.
Synthesis of 3-R-1,1-tetramethylene-2,3,4,4,5,10b-hexahydro-
1-chromeno[3,4-c]pyridine-2,4,5-triones through the Reformatsky reaction

175

Shelyakin V.V., Kartsev V.G., Yaremenko A.G., Lozinskii M.O.
Tandem reactions for modification of natural compounds

176

Shikhaliev Kh.S., Gusakova N.V., Shestakov A.S.
Reaction of 4,6-dimethyl-2-pyrimidinylhydrazine with derivatives of
2-ethoxymethylenemalonic acid

177

Silaichev P.S., Stepanyan Yu.G., Shchepin V.V.
Aryl 4-aryl-5-cyano-1-R-2,6-dioxopiperidine-3-carboxylates: Synthesis and reaction with amines

178

Silaichev P.S., Stepanyan Yu.G., Shchepin V.V.
Esters and amides of 2-R-1,3,4-trioxo-2,3-dihydro-1,9b-5-oxa-
2-aza-cyclopenta[2,3]cyclopropa[1,2-a]naphthalene-9-carboxylic acids

179

Silaichev P.S., Stepanyan Yu.G., Shchepin V.V.
3-Substituted alkyl 6-aryl-2,4-dioxo-5-cyano-3-aza-bicyclo[3,1,0]hexane-
1-carboxylates: Synthesis and reaction with amines

180

Silaichev P.S., Stepanyan Yu.G., Shchepin V.V.
5-Alkyl-6-aryl-3-R-2,4-dioxo-1-cyano-3-aza-bicyclo[3,1,0]hexanes

181

Slabko O.Yu., Kachanov A.V., Kaminskii V.A.
New electrophilic reactions of tetrahydropyrido[1,2-a]benzimidazoles

182

Slivchuk S.R., Rusanov E.B., Brovarets V.S.
A convenient approach to 7-substituted 3-arylsulfonylpyrazolo-
[1,5-a]pyrimidines

183

Smolyar N.N., Yutilov Yu.M., Gres'ko S.V.
4-Amino-6(hetaryl)pyridazin-3-ones:
Synthesis and cardiovascular activity

184

Sokolova M.S., Tereshchuk S.P., Gornostaev L.M.
Transformations of 1-acylamino-9,10-anthraquinone and 2-acylamino-
1,4-naphthoquinones

185

Sorotskaya L.N., Nevolina T.A., Krapivin G.D.
Hydroxamic acids based on 5-R-furfurylidene-5(4H)-oxazolones:
Synthesis and some reactions

186

Strakova I., Strakovs A., Petrova M., Belyakov S.
Nitrogen-containing 3,4-heteroannelated and 3-hetaryl-substituted coumarins

187

Sukach V.A., Bol'but A.V., Vovk M.V.
New polyfunctional 3,4-dihydropyrimidin-2(1)-ones

188

Sukhotin A.V., Kartsev V.G.
Substituted 2,3,4,5-tetrahydro-1H-1,5-benzodiazepin-2-ones

189

Sukhotin A.V., Kartsev V.G., Aleksandrov Yu.A.
Amino acids bearing a tetrahydropyrrole moiety

190

Takibaeva .., Ibraev .K., Kzhina Zh.., Gazaliev ..,
Nurkenov .., Kazerbaeva B.D.

Synthesis of 3-(1-p-nitrophenylethanol-2-yl)oxazolidine-2-thione

191

Tarabara I.N., Bondarenko Ya.S., Kas'yan L.I.
(9-Aryl-3,5-dioxo-4,9-diazatricyclo[5,3,1,08,10,02,6]undecan-4-yl)carboxylic acids: Synthesis and properties

192

Teterina N.M., Makhova T.V., Samartseva N.N., Yunnikova L.P., Makhmudov R.R., Bilevich I.O.
N-Arylmethylanilines containing N,O,S-heterocyclic moieties: Synthesis
and antimicrobial activity

193

Tkachenko Yu.N., Tsupak E.B.
Purino[8',7':2,3]imidazo[5,1-a]isoquinoline-10,12(9H,11H)-diones: Synthesis and reactivity

194

Tkachuk T.M., Pivovarenko V.G.
Azaheterocycles based on flavonoid glycosides

195

Tolkunov S.V., Kibal'nyi .V., Kryuchkov .., Afonin .., Dulenko V.I.
a-3-Chloropropylpyrilium salts in synthesis
of N-containing heterocycles

196

Tolkunov V.S., Dulenko V.I.
Synthesis of 5-hetero[2,3-e]diazepin-4-ones

197

Trofimov B.A., Petrova O.V., Ushakov I.A., Sobenina L.N., Mikhaleva A.I.
2-(1-Hydroxy-2,2-dicyanoethenyl)-1-methyl-4,5,6,7-tetrahydroindole: Synthesis and unusual rearrangement

198

Trostina A.V., Borisova T.N., Levov A.N., Voskressensky L.G.
Substituted tetrahydroazocino[4,5-b]indoles

199

Tsupak E.B., Tkachenko Yu.N.
Pyrrolo[3,2-d]pyrimidine-2,4-diones: Nitration and reduction to amines

200

Turmukhambetov A.Zh.,Burdel'naya E.V., Mukusheva G.K.,
Agedilova .., Kazantsev A.V., Adekenov S.., Shults E.E.

Reaction of alkaloids with tetramethylammonium iodide

201

Ulomskii E.N., Shestakova T.S., Deev S.L., Rusinov V.L., Chupakhin O.N.
New method for synthesis of Lamotridgine and other 3,5-diamino-
1,2,4-triazine derivatives

202

Usol'tseva N.V., Bykova V.V., Kudrik E.V., Anan'eva G.A.,
Zharnikova N.V., Shishkin V.N.

Induction of mesomorphic state in non-mesomorphic porphyrazine derivatives

203

Vasil'ev N.V., Romanov D.V., Truskanova T.D., Bazhenov ..,
Zatonskii G.V.

New cycloaddition reactions of 2,5-bis(perfluoroalkyl)-1,3,4-oxadiazoles

204

Vdovina S.V., Mamedov V.A., Mustakimova L.V., Gubaidullin A.T.,
Saifina A.F., Litvinov I.A., Reznik V.S.

Chelate compounds containing 3,4-dihydropyrimidin-2(1)-ne moieties

205

Velikorodov A.V., Imasheva N.M.
New carbamate derivatives of 1,4-benzoxazine

206

Velikorodov .V., Kovalev V.B., Borisov A.M., Kamanina N.A.
N,N'-Dimethoxycarbonyl-p-benzoquinonediimine in synthesis of carbamate derivatives of indole through the Nenitzescu reaction

207

Velikorodov .V., Kovalev V.B., Nagornaya Yu.V., Timchenko .V.
1,3-Dipolar cycloaddition of arenecarbonitrile N-oxides to -nitroso derivatives of N-arylcarbamates

208

Vikrishchuk N.I., Suvorova L.Yu., Popov L.D., Vikrishchuk A.D.
Arylvinyl- and hetarylvinyl-substituted 1,2,4-triazoles: Synthesis and alkylation

209

Vinogradova V.I., Zhurakulov Sh.N., Bobobekova D., Alimova M., Rakhimov Sh.B.
Derivatives of 1-phenyl-1,2,3,4,-tetrahydroisoquinoline

210

Vishnevskii Yu.V., Vilkov L.V., Ivanov A.A., Kuznetsov V.V.,
Makhova N.N.

Equilibrium geometry of N-chlorosuccinimide

211

Vydzhak R.N., Panchishin S.Ya., Kartsev V.G.
Polycyclic derivatives of pyrido[1,2-a]pyrimidine

212

Vypova N.L., Kazantseva D.S., Rakhimov Sh.B., Vinogradova V.I.
N-benzyl derivatives of cytisine: Hemostatic activity

213

Yamashkin S.A., Oreshkina E.A., Romanova I.S.
Pyrrolo[2,3-h]quinolines from 2,3-dimethyl- and 1,2,3-trimethyl-
4-aminoindoles

214

Yamashkin S.A., Zhukova N.V., Romanova I.S.
Reaction of 2,3-dimethyl- and 1,2,3-trimethyl-7-aminoindoles with oxalate

215

Yaremenko .G., Shelyakin V.V., Lozinskii ..
ulticomponent synthesis of new N,S-heterocyclic analogs of steroids

216

Yudashkin A.V., Golovin E.V.
Thermolysis of C-thienyl- and C-selenophenyltetrazoles

217

Yutilov Yu.M., Smolyar N.N., Svertilova I.A., Gres'ko C.V., Lomov D.A.
Condensed 6-methylpyridazin-3-ones

218

Zheldakova .., Rubinov D.B., Rubinova I.L.
Benzimidazole derivatives from alkoximes of cyclohexane b-triketones

219

Zhukovskaya .N., Anisimova V.., Spasov .., Chernikov .V.,
Yakovlev D.S.

Antiserotonin activity of 2-dialkylaminobenzimidazoles

220

Zhukovskaya .N., Anisimova V.., Spasov .., Kosolapov V.A.,
Chernikov .V., Naumenko L.V.

Biological activity of 2-benzylaminobenzimidazoles

221

Zicane D., Ravina I., Tetere Z., Petrova M.
3-Acylhexenylamido-1,2-dihydroquinazolin-4(3H)-ones from monohydrazides of cyclohexenedicarboxylic acids

222

Zorina A.V., Peshkov M.D., Shikhaliev Kh.S.
New heterocyclic systems by recyclizaition of arylmaleimides with
N,N-binucleophiles

223

Zubenko A.A., Fetisov L.N., Zubenko I.V., Sayapina E.A.
1,2,4-Triazolo[3,4-a]phthalazines: Synthesis and bioactivity


Friday, June 23, 2006

08:0009:00 Breakfast


Session I Chemistry of synthetic and natural heterocycles
(The Assembly Hall, the Big Reception-Room)


Oral Presentations

Session Chairpersons: Prof. Gy. Hajós, Prof. E. van der Eycken

9:009:15
Volochnyuk D.M., Pushechnikov A.O., Pinchuk A.M.,
Tolmachev A.A.
(Ukraine)
Fused 1,5,2-diaza- and 1,5,2-oxazaphosphinines: Synthesis and properties
9:159:30
Ol'shevskaya V.A., Zaitsev A.V., Savchenko A.N., Luzgina V.N., Shtil' A.A., Kalinin V.N. (Russia)
Carboranylporphyrins: Synthesis and bioactivity
9:309:45
Ershov A.Yu., Lagoda I.V., Koshmina N.V., Dobrodumov A.V. (Russia)
Recyclization of isoxazole derivatives
9:4510:00
Plaskon' A.S., Ryabukhin S.V., Volochnyuk D.M., Tolmachev A.A. (Ukraine)
3-Formylchromones in recyclization with 1,3-CCN- and
1,3--binucleophiles
10:0010:15
Makarenko S.V., Berestovitskaya V.M., Sadikov K.D., Tafeenko V.A., Chernyshev I.V. (Russia)
Potentially bioactive 1,4-benzodiazinones and their heteroanalogs:
Synthesis and structure
10:1510:30
Medvedeva A.S., Demina M.M., Novokshonov V.V., Safronova L.P.,
Rulev A.Yu., Pavlov D.V., Mareev A.V., Afonin A.V.
(Russia)
Synthesis of azidomethyl-1-1,2,3-triazoles
10:3010:45
Akhmetova V.R., Nadyrgulova G.R., Khairullina R.R., Khafizova S.R., Kunakova R.V., Dzhemilev U.M. (Russia)
One-pot synthesis of novel N,S-containing heterocycles
10:4511:00
Mikhalev O.V., Tarasevich B.N., Fedyanin I.V., Il'ina I.G. (Russia)
Autocomplexes of nitroaryls with heterocycles: Synthesis and characterization

11:0011:30 Coffee Break (The Banquet Hall, the Big Reception-Room)

11:3013:30 (Lecture-Room 2, The Big Reception-Room)
Round table
       Moderator: Actagon AB, Stockholm, Sweden
       Participants: VIP delegates only (including heads of research centers, CEOs of companies and the mayor of the Chernogolovka Research Center)
       "Prospects for the development of international projects in biotechnology: realization and investment algorithms"


Session I Chemistry of synthetic and natural heterocycles
(Session For Russian and CIS Delegates. Working language is Russian)

(The Assembly Hall, the Big Reception-Room)


Oral Presentations

Session Chairpersons: Prof. A. Nemes, Prof. G. Danagulyan

11:3011:45
Popkov S.V., Kovalenko L.V. (Russia)
1-Azolylmethyl-6-benzylidene-2-alkoxy-2-methyl- and
2,2-dimethylcyclohexanols: Synthesis and bioactivity
11:4512:00
Przheval'skii N.M. (Russia)
Heterohexadiens in synthesis of heterocycles
12:0012:15
Samsoniya Sh.A., Trapaidze M.V., Gogrichiani E.O., Katsadze E.A., Maisuradze J.P., Dzhaparidze K.G. (Georgia)
Some spiro derivatives of indole and condensed bis-indoles
12:1512:30
Semenov V.E., Nikolaev A.E., Giniyatullin R.Kh., Lodochnikova O.A., Voloshina A.D., Galiullina L.F., Latypov Sh.K., Reznik V.S. (Russia)
Pyrimidinophanes with nitrogen atoms in bridging groups:
Synthesis and properties
12:3012:45
Isak A.D., Pogorelova I.P., Tyupalo N.F., Isak V.A. (Ukraine)
Pyrimidine sulfone amides and their derivatives: Synthesis and biological activity
12:4513:00
Sirakanyan S.N., Kartsev V.G., Paronikyan E.G., Noravyan A.S. (Armenia)
Derivatives of 2,7-naphthyridine: Synthesis, transformations, and bioactivity
13:0013:15
Shestakov A.S., Gusakova N.V., Shikhaliev Kh.S. (Russia)
Cyanamides and their derivatives in reactions of heterocyclyzation
13:1513:30
Paronikyan E.G., Noravyan A.S., Hakobyan Sh.F. (Armenia)
New condensed thieno[3,2-d]pyrimidines and thieno[3,2-d]-1,2,3-triazines: Synthesis and bioactivity
13:3013:45
Kovalenko S.N., Silin .V., Savchenko .I. (Ukraine)
Synthesis and reactivity of pyrazolo[4,3-c]quinolines


14:0016:00 Closing Ceremony and Champagne Party
16:00 Departure